日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

I‑GAT: Interpretable Graph Attention Networks for Ligand Optimization

I-GAT:用于配体优化的可解释图注意力网络

Mathew, Ezek; Emmitte, Kyle A; Liu, Jin

Developing inhibitors of the guanosine triphosphate hydrolysis accelerating activity of Regulator of G protein Signaling-14

开发鸟苷三磷酸水解加速G蛋白信号调节因子-14活性的抑制剂

Agogo-Mawuli, Percy S; Sadiya, Isra; Abramyan, Tigran M; Bosch, Dustin E; Emmitte, Kyle A; Colón-Pérez, Luis M; Kosloff, Mickey; Siderovski, David P

Efficient Regioselective Synthesis of Benzimidazoles and Azabenzimidazoles to Enable the Rapid Development of Structure-Activity Relationships for Activation of SLACK Potassium Channels

高效区域选择性合成苯并咪唑和氮杂苯并咪唑,以快速建立SLACK钾通道激活的构效关系

Peprah, Paul K; Spitznagel, Brittany D; Du, Yu; Nguyen, Dalena; Weaver, C David; Emmitte, Kyle A

Developing inhibitors of the guanosine triphosphate hydrolysis accelerating activity of Regulator of G protein Signaling-14

开发鸟苷三磷酸水解加速G蛋白信号调节因子-14活性的抑制剂

Agogo-Mawuli, Percy S; Sadiya, Isra; Abramyan, Tigran M; Bosch, Dustin E; Emmitte, Kyle A; Colon-Perez, Luis; Kosloff, Mickey; Siderovski, David P

Phenethylaminylation: Preliminary In Vitro Evidence for the Covalent Transamidation of Psychedelic Phenethylamines to Glial Proteins using 3,5-Dimethoxy-4-(2-Propynyloxy)-Phenethylamine as a Model Compound

苯乙胺化:以3,5-二甲氧基-4-(2-丙炔氧基)-苯乙胺为模型化合物,初步体外证据表明迷幻苯乙胺可共价转酰胺化为神经胶质蛋白。

Rangan, Rajiv S; Petty, R Max; Acharya, Suchismita; Emmitte, Kyle A; do Valle, Rafael S; Lam, Chandra; Essajee, Salman I; Mayhew, William; Young, Olivia; Brooks, Calvin D; Forster, Michael J; Tovar-Vidales, Tara; Clark, Abbot F

Heterozygous expression of a Kcnt1 gain-of-function variant has differential effects on somatostatin- and parvalbumin-expressing cortical GABAergic neurons

Kcnt1 功能获得性变异的杂合表达对表达生长抑素和小清蛋白的皮质 GABA 能神经元有不同的影响

Amy N Shore, Keyong Li, Mona Safari, Alshaima'a M Qunies, Brittany D Spitznagel, C David Weaver, Kyle Emmitte, Wayne Frankel, Matthew C Weston1

Heterozygous expression of a Kcnt1 gain-of-function variant has differential effects on SST- and PV-expressing cortical GABAergic neurons

Kcnt1功能获得性变异体的杂合表达对表达SST和PV的皮质GABA能神经元具有不同的影响

Shore, Amy N; Li, Keyong; Safari, Mona; Qunies, Alshaima'a M; Spitznagel, Brittany D; Weaver, C David; Emmitte, Kyle A; Frankel, Wayne N; Weston, Matthew C

Quercetin and Related Analogs as Therapeutics to Promote Tissue Repair

槲皮素及其类似物作为促进组织修复的治疗药物

McKay, Tina B; Emmitte, Kyle A; German, Carrie; Karamichos, Dimitrios

Structure-activity relationship studies in a new series of 2-amino-N-phenylacetamide inhibitors of Slack potassium channels

对一系列新型2-氨基-N-苯基乙酰胺类Slack钾通道抑制剂进行了构效关系研究

Qunies, Alshaima'a M; Mishra, Nigam M; Spitznagel, Brittany D; Du, Yu; Acuña, Valerie S; David Weaver, C; Emmitte, Kyle A

Small-molecule inhibitors of Slack potassium channels as potential therapeutics for childhood epilepsies

小分子Slack钾通道抑制剂作为治疗儿童癫痫的潜在药物

M Qunies, Alshaima'a; A Emmitte, Kyle