日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Native Taylor/Non-Taylor Dispersion-Mass Spectrometry (TNT-MS) Allows Rapid Protein Desalting and Multiplexed, Label-Free Ligand Screening

原生泰勒/非泰勒色散质谱(TNT-MS)可实现快速蛋白质脱盐和多重无标记配体筛选

Eisert, Jonathan; Maciel, Edvaldo Vasconcelos Soares; Dederer, Verena; Berwanger, Aylin; Bailey, Henry J; Đikić, Ivan; Knapp, Stefan; Empting, Martin; Mathea, Sebastian; Jensen, Henrik; Lermyte, Frederik

Th17 cells favor migration and invasiveness of cervical cancer cells under hypoxia in an IGF2BP2-dependent manner

Th17细胞以IGF2BP2依赖的方式促进缺氧条件下宫颈癌细胞的迁移和侵袭。

Gies, Selina; Pohlers, Maike; Tänzer, Tanja; Ampofo, Emmanuel; Laschke, Matthias W; Schäfer, Moritz; Kim, Yoo-Jin; Bohle, Rainer Maria; Solomayer, Erich-Franz; Wagner, Konrad; Empting, Martin; Kiemer, Alexandra K; Walch-Rückheim, Barbara

Toward Anti-Herpesviral PROTACs: Assessing the Challenges for Targeted Protein Degradation on the Example of Kaposi's Sarcoma-Associated Herpesvirus Latency-Associated Nuclear Antigen

迈向抗疱疹病毒PROTAC:以卡波西肉瘤相关疱疹病毒潜伏相关核抗原为例评估靶向蛋白降解的挑战

Berwanger, Aylin; Stein, Saskia Catherina; Brandner, Sarah; Kany, Andreas Martin; Heinz, Sebastian; Loretz, Brigitta; Lehr, Claus-Michael; Hirsch, Anna Katharina Herta; Lermyte, Frederik; Schulz, Thomas Friedrich; Empting, Martin

Identification of targetable vulnerabilities of PLK1-overexpressing cancers by synthetic dosage lethality.

通过合成剂量致死性鉴定 PLK1 过表达癌症的可靶向脆弱性

Cunningham Chelsea E, Vizeacoumar Frederick S, Zhang Yue, Kyrylenko Liliia, Both Simon, Maranda Vincent, Dong He, Price Jared D W, Gao Peng, Wagner Konrad, Wu Yingwen, Lazell-Wright Mary, Ganapathysamy Ashtalakshmi, Hari Rithik, Bhanumathy Kalpana K, Denomy Connor, Saxena Anjali, Vizeacoumar Jeff P, Morales Alain Morejon, Khan Faizaan, Mosley Shayla, Chen Angie, Katrii Tetiana, Zoller Ben G E, Rajamanickam Karthic, Walke Prachi, Gong Lihui, Patel Hardikkumar, Elhasasna Hussain, Dahiya Renuka, Abuhussein Omar, Dmitriev Anton, Freywald Tanya, Munhoz Erika Prando, Ruppin Eytan, Lee Joo Sang, Rox Katharina, Koebel Martin, Hopkins Laura, Lee Cheng Han, Yadav Sunil, Gasparoni Gilles, Walter Jörn, Krishnan Anand, Datla Raju, Toosi Behzad, Baker Kristi, Meens Jalna, Cescon David W, Ailles Laurie, Leary Scot C, Wu Yuliang, Empting Martin, Kiemer Alexandra K, Freywald Andrew, Vizeacoumar Franco J

Domain adaptable language modeling of chemical compounds identifies potent pathoblockers for Pseudomonas aeruginosa

化学化合物的领域自适应语言建模可识别出铜绿假单胞菌的有效致病阻断剂

Kallergis, Georgios; Asgari, Ehsannedin; Empting, Martin; Hirsch, Anna K H; Klawonn, Frank; McHardy, Alice C

Nanoparticles in liposomes: a platform for increased antibiotic selectivity in multidrug resistant bacteria in respiratory tract infections.

脂质体中的纳米颗粒:提高呼吸道感染中多重耐药菌抗生素选择性的平台

Fakhoury Nathalie E, Mansour Samar, Abdel-Halim Mohammad, Hamed Mostafa M, Empting Martin, Boese Annette, Loretz Brigitta, Lehr Claus-Michael, Tammam Salma N

Enzyme-Linked Lipid Nanocarriers for Coping Pseudomonal Pulmonary Infection. Would Nanocarriers Complement Biofilm Disruption or Pave Its Road?

酶联脂质纳米载体在应对铜绿假单胞菌肺部感染中的应用:纳米载体是辅助生物膜破坏还是为其铺平道路?

Nafee, Noha; Gaber, Dina M; Abouelfetouh, Alaa; Alseqely, Mustafa; Empting, Martin; Schneider, Marc

Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof-of-Principle

PqsR反向激动剂转化研究进展:从体外功效优化到体内原理验证

Hamed, Mostafa M; Abdelsamie, Ahmed S; Rox, Katharina; Schütz, Christian; Kany, Andreas M; Röhrig, Teresa; Schmelz, Stefan; Blankenfeldt, Wulf; Arce-Rodriguez, Alejandro; Borrero-de Acuña, José Manuel; Jahn, Dieter; Rademacher, Jessica; Ringshausen, Felix C; Cramer, Nina; Tümmler, Burkhard; Hirsch, Anna K H; Hartmann, Rolf W; Empting, Martin

Towards the sustainable discovery and development of new antibiotics

迈向新型抗生素的可持续发现和开发

Miethke, Marcus; Pieroni, Marco; Weber, Tilmann; Brönstrup, Mark; Hammann, Peter; Halby, Ludovic; Arimondo, Paola B; Glaser, Philippe; Aigle, Bertrand; Bode, Helge B; Moreira, Rui; Li, Yanyan; Luzhetskyy, Andriy; Medema, Marnix H; Pernodet, Jean-Luc; Stadler, Marc; Tormo, José Rubén; Genilloud, Olga; Truman, Andrew W; Weissman, Kira J; Takano, Eriko; Sabatini, Stefano; Stegmann, Evi; Brötz-Oesterhelt, Heike; Wohlleben, Wolfgang; Seemann, Myriam; Empting, Martin; Hirsch, Anna K H; Loretz, Brigitta; Lehr, Claus-Michael; Titz, Alexander; Herrmann, Jennifer; Jaeger, Timo; Alt, Silke; Hesterkamp, Thomas; Winterhalter, Mathias; Schiefer, Andrea; Pfarr, Kenneth; Hoerauf, Achim; Graz, Heather; Graz, Michael; Lindvall, Mika; Ramurthy, Savithri; Karlén, Anders; van Dongen, Maarten; Petkovic, Hrvoje; Keller, Andreas; Peyrane, Frédéric; Donadio, Stefano; Fraisse, Laurent; Piddock, Laura J V; Gilbert, Ian H; Moser, Heinz E; Müller, Rolf

Squalenyl Hydrogen Sulfate Nanoparticles for Simultaneous Delivery of Tobramycin and an Alkylquinolone Quorum Sensing Inhibitor Enable the Eradication of P. aeruginosa Biofilm Infections

角鲨烯基硫酸氢盐纳米颗粒可同时递送妥布霉素和烷基喹诺酮类群体感应抑制剂,从而根除铜绿假单胞菌生物膜感染

Ho, Duy-Khiet; Murgia, Xabier; De Rossi, Chiara; Christmann, Rebekka; Hüfner de Mello Martins, Antonio G; Koch, Marcus; Andreas, Anastasia; Herrmann, Jennifer; Müller, Rolf; Empting, Martin; Hartmann, Rolf W; Desmaele, Didier; Loretz, Brigitta; Couvreur, Patrick; Lehr, Claus-Michael