日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Design of New Series of Sulfonates with Potent and Specific BChE Inhibition and Anti-Inflammatory Effects

基于结构的新型磺酸盐系列设计及其强效和特异性的丁酰胆碱酯酶抑制和抗炎作用

Kurma, Siva Hariprasad; Adarvez-Feresin, Camila; Parravicini, Oscar; Garro, Adriana; Stepankova, Sarka; Hosek, Jan; Pauk, Karel; Lisicic, Jovana; Jampilek, Josef; Enriz, Ricardo Daniel; Imramovsky, Ales

Integrated In Vitro and In Silico Profiling of Piperazinyl Thiosemicarbazone Derivatives Against Trypanosoma cruzi: Stage-Specific Activity and Enzyme Inhibition

哌嗪基硫代氨基脲衍生物抗克氏锥虫活性的体外和计算机模拟综合分析:阶段特异性活性和酶抑制

Baldoni, Héctor A; Sbaraglini, María L; Balcazar, Darío E; Arias, Diego G; Guerrero, Sergio A; Alba Soto, Catalina D; Cieslik, Wioleta; Rogalska, Marta; Polański, Jaroslaw; Enriz, Ricardo D; Jampilek, Josef; Musiol, Robert

Rosmarinic Acid Present in Lepechinia floribunda and Lepechinia meyenii as a Potent Inhibitor of the Adenylyl Cyclase gNC1 from Giardia lamblia

迷迭香酸存在于 Lepechinia floribunda 和 Lepechinia meyenii 中,是贾第鞭毛虫腺苷酸环化酶 gNC1 的强效抑制剂。

Zurita, Adolfo; Vega Hissi, Esteban; Cianci Romero, Agostina; Luján, Adela María; Salido, Sofía; Yaneff, Agustín; Davio, Carlos; Cobo, Justo; Carpinella, María Cecilia; Enriz, Ricardo Daniel

New ATP-competitive inhibitors of E. coli GyrB obtained from the mapping of the hydrophobic floor at the binding site: synthesis and biological evaluation

通过对结合位点疏水表面的映射获得大肠杆菌 GyrB 的新型 ATP 竞争性抑制剂:合成与生物学评价

Lucas Gutierrez, Peter Peršolja, Rodrigo Tosso, Nace Zidar, Danijel Kikelj, Ricardo D Enriz

Arylated analogues of cypronazole: fungicidal effect and activity on human fibroblasts. Docking analysis and molecular dynamics simulations

环丙唑醇芳基化类似物:杀菌作用及对人成纤维细胞的活性。分子对接分析和分子动力学模拟

Herrera Cano, Natividad; Andujar, Sebastian A; Theoduloz, Cristina; Wunderlin, Daniel A; Santiago, Ana N; Schmeda-Hirschmann, Guillermo; Enriz, Ricardo D; Feresin, Gabriela E

Novel Sulfonamide-Based Carbamates as Selective Inhibitors of BChE

新型磺酰胺基氨基甲酸酯作为 BChE 的选择性抑制剂

Pratibha Magar, Oscar Parravicini, Šárka Štěpánková, Katarina Svrčková, Adriana D Garro, Izabela Jendrzejewska, Karel Pauk, Jan Hošek, Josef Jampílek, Ricardo D Enriz, Aleš Imramovský

Design of new quinolin-2-one-pyrimidine hybrids as sphingosine kinases inhibitors

设计新型喹啉-2-酮-嘧啶杂合物作为鞘氨醇激酶抑制剂

Vettorazzi, Marcela; Insuasty, Daniel; Lima, Santiago; Gutiérrez, Lucas; Nogueras, Manuel; Marchal, Antonio; Abonia, Rodrigo; Andújar, Sebastián; Spiegel, Sarah; Cobo, Justo; Enriz, Ricardo D

Arylaminopropanone Derivatives as Potential Cholinesterase Inhibitors: Synthesis, Docking Study and Biological Evaluation

芳氨基丙酮衍生物作为潜在胆碱酯酶抑制剂的合成、对接研究及生物评价

Anna Hudcová, Aleš Kroutil, Renata Kubínová, Adriana D Garro, Lucas J Gutierrez, Daniel Enriz, Michal Oravec, Jozef Csöllei

Targeting defective sphingosine kinase 1 in Niemann-Pick type C disease with an activator mitigates cholesterol accumulation

利用激活剂靶向尼曼匹克 C 型疾病中缺陷的鞘氨醇激酶 1 可减轻胆固醇的积累

Jason Newton, Elisa N D Palladino, Cynthia Weigel, Michael Maceyka, Markus H Gräler, Can E Senkal, Ricardo D Enriz, Pavlina Marvanova, Josef Jampilek, Santiago Lima, Sheldon Milstien, Sarah Spiegel

Small Cationic Peptides: Influence of Charge on Their Antimicrobial Activity

小阳离子肽:电荷对其抗菌活性的影响

López Cascales, José Javier; Zenak, Siham; García de la Torre, José; Lezama, Osvaldo Guy; Garro, Adriana; Enriz, Ricardo Daniel