日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Distal protein-protein interactions contribute to nirmatrelvir resistance

远端蛋白质-蛋白质相互作用导致尼尔马特雷韦耐药性

Eric M Lewandowski # ,Xiujun Zhang # ,Haozhou Tan # ,Aiden Jaskolka-Brown ,Navita Kohaal ,Aliaksandra Frazier ,Jesper J Madsen ,Lian M C Jacobs ,Jun Wang ,Yu Chen

Naturally Occurring Mutations of SARS-CoV-2 Main Protease Confer Drug Resistance to Nirmatrelvir

SARS-CoV-2 主蛋白酶的自然突变赋予其对尼马替利韦的耐药性

Yanmei Hu ,Eric M Lewandowski ,Haozhou Tan ,Xiaoming Zhang ,Ryan T Morgan ,Xiujun Zhang ,Lian M C Jacobs ,Shane G Butler ,Maura V Gongora ,John Choy ,Xufang Deng ,Yu Chen ,Jun Wang

A yeast-based system to study SARS-CoV-2 M pro structure and to identify nirmatrelvir resistant mutations

基于酵母的系统研究 SARS-CoV-2 M pro 结构并识别尼玛瑞韦耐药突变

Jin Ou, Eric M Lewandowski, Yanmei Hu, Austin A Lipinski, Ryan T Morgan, Lian M C Jacobs, Xiujun Zhang, Melissa J Bikowitz, Paul Langlais, Haozhou Tan, Jun Wang, Yu Chen, John S Choy

Naturally occurring mutations of SARS-CoV-2 main protease confer drug resistance to nirmatrelvir

SARS-CoV-2 主要蛋白酶的自然突变导致尼玛瑞韦产生耐药性

Yanmei Hu, Eric M Lewandowski, Haozhou Tan, Xiaoming Zhang, Ryan T Morgan, Xiujun Zhang, Lian M C Jacobs, Shane G Butler, Maura V Gongora, John Choy, Xufang Deng, Yu Chen, Jun Wang

Differential long-term regulation of TAS2R14 by structurally distinct agonists

结构不同的激动剂对 TAS2R14 的差异化长期调节

Jung A Woo, Maria Castaño, Ashley Goss, Donghwa Kim, Eric M Lewandowski, Yu Chen, Stephen B Liggett

Structural and Mechanistic Analysis of Drosophila melanogaster Agmatine N-Acetyltransferase, an Enzyme that Catalyzes the Formation of N-Acetylagmatine

果蝇胍丁胺 N-乙酰转移酶(一种催化 N-乙酰胍丁胺形成的酶)的结构和机制分析

Daniel R Dempsey, Derek A Nichols, Matthew R Battistini, Orville Pemberton, Santiago Rodriguez Ospina, Xiujun Zhang, Anne-Marie Carpenter, Brian G O'Flynn, James W Leahy, Ankush Kanwar, Eric M Lewandowski, Yu Chen, David J Merkler