日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Melanocortin 3 receptor regulates hepatic autophagy and systemic adiposity.

黑皮质素 3 受体调节肝脏自噬和全身脂肪沉积

Patel Tushar P, Jun Joo Yun, Seo Arnold Y, Levi Noah J, Elizondo Diana M, Chen Jocelyn, Wong Adrian M, Tugarinov Nicol, Altman Elizabeth K, Gehle Daniel B, Jung Sun Min, Patel Pooja, Ericson Mark, Haskell-Luevano Carrie, Demby Tamar C, Cougnoux Antony, Wolska Anna, Yanovski Jack A

N-Branched Tricyclic Guanidines as Novel Melanocortin-3 Receptor Agonists and Melanocortin-4 Receptor Antagonists

N-支链三环胍类化合物作为新型黑皮质素-3受体激动剂和黑皮质素-4受体拮抗剂

Weirath, Nicholas A; Zajac, Jonathan W P; Donow, Haley M; Lavoi, Travis M; Pinilla, Clemencia; Santos, Radleigh G; Prajapati, Ritu; Speth, Robert; Ericson, Mark D; Sarupria, Sapna; Giulianotti, Marcello A; Haskell-Luevano, Carrie

Rare variants in the melanocortin 4 receptor gene (MC4R) are associated with abdominal fat and insulin resistance in youth with obesity

黑皮质素4受体基因(MC4R)的罕见变异与肥胖青少年的腹部脂肪堆积和胰岛素抵抗有关。

Galuppo, Brittany; Mannam, Prabhath; Bonet, Jacopo; Pierpont, Bridget; Trico', Domenico; Haskell-Luevano, Carrie; Ericson, Mark D; Freeman, Katie T; Philbrick, William M; Bale, Allen E; Caprio, Sonia; Santoro, Nicola

Incorporation of Indoylated Phenylalanine Yields a Sub-Micromolar Selective Melanocortin-4 Receptor Antagonist Tetrapeptide

掺入吲哚基苯丙氨酸可得到亚微摩尔级选择性黑皮质素-4受体拮抗剂四肽。

Ericson, Mark D; Larson, Courtney M; Freeman, Katie T; Nicke, Lennart; Geyer, Armin; Haskell-Luevano, Carrie

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput "Unbiased" Screening Campaign

通过高通量“无偏”筛选活动发现纳摩尔级黑素皮质素-3受体(MC3R)选择性小分子吡咯烷双环胍激动剂化合物

Doering, Skye R; Freeman, Katie; Debevec, Ginamarie; Geer, Phaedra; Santos, Radleigh G; Lavoi, Travis M; Giulianotti, Marc A; Pinilla, Clemencia; Appel, Jon R; Houghten, Richard A; Ericson, Mark D; Haskell-Luevano, Carrie

The melanocortin pathway and energy homeostasis: From discovery to obesity therapy

黑皮质素通路与能量稳态:从发现到肥胖治疗

Yeo, Giles S H; Chao, Daniela Herrera Moro; Siegert, Anna-Maria; Koerperich, Zoe M; Ericson, Mark D; Simonds, Stephanie E; Larson, Courtney M; Luquet, Serge; Clarke, Iain; Sharma, Shubh; Clément, Karine; Cowley, Michael A; Haskell-Luevano, Carrie; Van Der Ploeg, Lex; Adan, Roger A H

Human β-Defensin 1 and β-Defensin 3 (Mouse Ortholog mBD14) Function as Full Endogenous Agonists at Select Melanocortin Receptors

人β-防御素1和β-防御素3(小鼠同源物mBD14)在特定黑皮质素受体上发挥完全内源性激动剂的作用

Ericson, Mark D; Singh, Anamika; Tala, Srinivasa R; Haslach, Erica M; Dirain, Marvin L S; Schaub, Jay W; Flores, Viktor; Eick, Natalie; Lensing, Cody J; Freeman, Katie T; Smeester, Branden A; Adank, Danielle N; Wilber, Stacey L; Speth, Robert; Haskell-Luevano, Carrie

A Review of Single-Nucleotide Polymorphisms in Orexigenic Neuropeptides Targeting G Protein-Coupled Receptors

对靶向G蛋白偶联受体的促食神经肽中的单核苷酸多态性进行综述

Ericson, Mark D; Haskell-Luevano, Carrie

Bench-top to clinical therapies: A review of melanocortin ligands from 1954 to 2016

从实验室研究到临床治疗:1954年至2016年黑皮质素配体的回顾

Ericson, Mark D; Lensing, Cody J; Fleming, Katlyn A; Schlasner, Katherine N; Doering, Skye R; Haskell-Luevano, Carrie

A fragment of the Escherichia coli ClpB heat-shock protein is a micromolar melanocortin 1 receptor agonist

大肠杆菌ClpB热休克蛋白的一个片段是微摩尔级的黑皮质素1受体激动剂。

Ericson, Mark D; Schnell, Sathya M; Freeman, Katie T; Haskell-Luevano, Carrie