Targeting interleukin-2-inducible T-cell kinase (ITK) and resting lymphocyte kinase (RLK) using a novel covalent inhibitor PRN694
使用新型共价抑制剂 PRN694 靶向白细胞介素 2 诱导 T 细胞激酶 (ITK) 和静息淋巴细胞激酶 (RLK)
期刊:Journal of Biological Chemistry
影响因子:4
doi:10.1074/jbc.M114.614891
Yiming Zhong, Shuai Dong, Ethan Strattan, Li Ren, Jonathan P Butchar, Kelsey Thornton, Anjali Mishra, Pierluigi Porcu, J Michael Bradshaw, Angelina Bisconte, Timothy D Owens, Erik Verner, Ken A Brameld, Jens Oliver Funk, Ronald J Hill, Amy J Johnson, Jason A Dubovsky