日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of a Highly Cooperative PROTAC Degrader Targeting GTP-Loaded KRAS(On) Alleles

鉴定一种高度协同的PROTAC降解酶,该酶靶向GTP结合的KRAS(On)等位基因

Vetma, Vesna; Puoti, Ilaria; Karolak, Natalia K; Chakraborti, Sohini; Diers, Emelyne; Girardi, Enrico; Khan, Shakil; Kidd, Giorgia; Kropatsch, Katrin G; Mclennan, Ross; O'Connor, Suzanne; Samwer, Matthias; Trainor, Nicole; Whitworth, Claire; Wijaya, Andre J; Wong, Jeff Y F; Zollman, David; Farnaby, William; Popow, Johannes; Ciulli, Alessio; Ettmayer, Peter; McAulay, Kirsten

Chasing Red Herrings: Palladium Metal Salt Impurities Feigning KRAS Activity in Biochemical Assays.

追逐虚假信号:钯金属盐杂质在生化测定中伪装成 KRAS 活性

Gerstberger Thomas, Berger Helmut, Büttner Frank H, Gmachl Michael, Kessler Dirk, Koegl Manfred, Lucas Simon, Martin Laetitia J, Mayer Moriz, McConnell Darryl B, Mitzner Sophie, Scholz Guido, Treu Matthias, Wolkerstorfer Bernhard, Zahn Stephan, Zak Krzysztof M, Jaeger Philipp A, Ettmayer Peter

In-vitro effects of novel periodontal scalers with a planar ultrasonic piezoelectric transducer on periodontal biofilm removal, dentine surface roughness, and periodontal ligament fibroblasts adhesion

新型平面超声压电换能器牙周刮治器对牙周生物膜去除、牙本质表面粗糙度和牙周膜成纤维细胞粘附的体外影响

Berto, Luciana Aranha; Ettmayer, Johanna Blanda; Stutzer, Diego; Nietzsche, Sandor; Niederhauser, Thomas; Burger, Juergen; Sculean, Anton; Eick, Sigrun; Hofmann, Martin

BI-3406, a Potent and Selective SOS1-KRAS Interaction Inhibitor, Is Effective in KRAS-Driven Cancers through Combined MEK Inhibition

BI-3406 是一种强效且选择性的 SOS1-KRAS 相互作用抑制剂,可通过联合 MEK 抑制有效治疗 KRAS 驱动的癌症

Marco H Hofmann #, Michael Gmachl #, Juergen Ramharter #, Fabio Savarese, Daniel Gerlach, Joseph R Marszalek, Michael P Sanderson, Dirk Kessler, Francesca Trapani, Heribert Arnhof, Klaus Rumpel, Dana-Adriana Botesteanu, Peter Ettmayer, Thomas Gerstberger, Christiane Kofink, Tobias Wunberg, Andreas Z

The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification

激酶化学基因组学数据集(KCGS):用于识别激酶脆弱性的开放科学资源

Wells, Carrow I; Al-Ali, Hassan; Andrews, David M; Asquith, Christopher R M; Axtman, Alison D; Dikic, Ivan; Ebner, Daniel; Ettmayer, Peter; Fischer, Christian; Frederiksen, Mathias; Futrell, Robert E; Gray, Nathanael S; Hatch, Stephanie B; Knapp, Stefan; Lücking, Ulrich; Michaelides, Michael; Mills, Caitlin E; Müller, Susanne; Owen, Dafydd; Picado, Alfredo; Saikatendu, Kumar S; Schröder, Martin; Stolz, Alexandra; Tellechea, Mariana; Turunen, Brandon J; Vilar, Santiago; Wang, Jinhua; Zuercher, William J; Willson, Timothy M; Drewry, David H

Native Mass Spectrometry Can Effectively Predict PROTAC Efficacy

天然质谱法可有效预测 PROTAC 功效

Rebecca Beveridge, Dirk Kessler, Klaus Rumpel, Peter Ettmayer, Anton Meinhart, Tim Clausen

Progress towards a public chemogenomic set for protein kinases and a call for contributions

构建蛋白质激酶公共化学基因组数据集的进展及贡献征集

Drewry, David H; Wells, Carrow I; Andrews, David M; Angell, Richard; Al-Ali, Hassan; Axtman, Alison D; Capuzzi, Stephen J; Elkins, Jonathan M; Ettmayer, Peter; Frederiksen, Mathias; Gileadi, Opher; Gray, Nathanael; Hooper, Alice; Knapp, Stefan; Laufer, Stefan; Luecking, Ulrich; Michaelides, Michael; Müller, Susanne; Muratov, Eugene; Denny, R Aldrin; Saikatendu, Kumar S; Treiber, Daniel K; Zuercher, William J; Willson, Timothy M