日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of Orthosteric GABA(B) Receptor Ligands by Virtual Screening and In Vitro Validation.

通过虚拟筛选和体外验证鉴定正构GABA(B)受体配体

Evenseth Linn S M, Russotto Clizia, Wushur Imin, Warszycki Dawid, Moldes-Anaya Angel S, Bojarski Andrzej J, Gabrielsen Mari, Sylte Ingebrigt

Exploring Conformational Dynamics of the Extracellular Venus flytrap Domain of the GABA(B) Receptor: A Path-Metadynamics Study

探索GABA(B)受体胞外维纳斯捕蝇草结构域的构象动力学:一项路径元动力学研究

Evenseth, Linn S M; Ocello, Riccardo; Gabrielsen, Mari; Masetti, Matteo; Recanatini, Maurizio; Sylte, Ingebrigt; Cavalli, Andrea

The GABA(B) Receptor-Structure, Ligand Binding and Drug Development

GABA(B)受体——结构、配体结合和药物开发

Evenseth, Linn Samira Mari; Gabrielsen, Mari; Sylte, Ingebrigt

In Silico Methods for the Discovery of Orthosteric GABA(B) Receptor Compounds

利用计算机模拟方法发现正构GABA(B)受体化合物

Evenseth, Linn M; Warszycki, Dawid; Bojarski, Andrzej J; Gabrielsen, Mari; Sylte, Ingebrigt

Exploring the overlapping binding sites of ifenprodil and EVT-101 in GluN2B-containing NMDA receptors using novel chicken embryo forebrain cultures and molecular modeling

使用新型鸡胚前脑培养和分子建模探索艾芬地尔和 EVT-101 在含 GluN2B 的 NMDA 受体中的重叠结合位点

Marthe F Fjelldal, Thibaud Freyd, Linn M Evenseth, Ingebrigt Sylte, Avi Ring, Ragnhild E Paulsen

In Silico Site-Directed Mutagenesis Informs Species-Specific Predictions of Chemical Susceptibility Derived From the Sequence Alignment to Predict Across Species Susceptibility (SeqAPASS) Tool

利用计算机模拟定点诱变技术,结合序列比对预测跨物种化学敏感性(SeqAPASS)工具,可以对物种特异性化学敏感性进行预测。

Doering, Jon A; Lee, Sehan; Kristiansen, Kurt; Evenseth, Linn; Barron, Mace G; Sylte, Ingebrigt; LaLone, Carlie A