Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors
氧代吡啶并[2,3-d]嘧啶类化合物作为共价L858R/T790M突变选择性表皮生长因子受体(EGFR)抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5b00193
Wurz, Ryan P; Pettus, Liping H; Ashton, Kate; Brown, James; Chen, Jian Jeffrey; Herberich, Brad; Hong, Fang-Tsao; Hu-Harrington, Essa; Nguyen, Tom; St Jean, David J Jr; Tadesse, Seifu; Bauer, David; Kubryk, Michele; Zhan, Jinghui; Cooke, Keegan; Mitchell, Petia; Andrews, Kristin L; Hsieh, Faye; Hickman, Dean; Kalyanaraman, Nataraj; Wu, Tian; Reid, Darren L; Lobenhofer, Edward K; Andrews, Dina A; Everds, Nancy; Guzman, Roberto; Parsons, Andrew T; Hedley, Simon J; Tedrow, Jason; Thiel, Oliver R; Potter, Matthew; Radinsky, Robert; Beltran, Pedro J; Tasker, Andrew S