日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Triazine-Based Toll-Like Receptor 9 Antagonists with Oral Activity

发现具有口服活性的三嗪类 Toll 样受体 9 拮抗剂

Mandler, Michael D; Zhu, Yeheng; Hollenbeck, Emily C; Ziegler, Milinda; Posy, Shana L; Mukundan, Shilpaa; Halpern, O Scott; Driscoll, James P; Wang, Tao; Huang, Li; Fernando, Gayani; Jung, Helen; Li, Ling; Cutrone, Jingfang; Baswar, Dnyaneshwar; Eapen, Prasanth; Traeger, Sarah C; Srivastava, Shivangi; Olsen, Jonathan; Everlof, Gerry G; Trujillo, Glenda; Ellsworth, Bruce A; Regueiro-Ren, Alicia

Balanced Permeability Index: A Multiparameter Index for Improved In Vitro Permeability

平衡渗透指数:一种用于改善体外渗透性的多参数指数

Weiss, Dahlia R; Baylon, Javier L; Evans, Ethan D; Paiva, Anthony; Everlof, Gerry; Cutrone, Jingfang; Broccatelli, Fabio

Antithrombotic Effects of Combined PAR (Protease-Activated Receptor)-4 Antagonism and Factor Xa Inhibition

PAR(蛋白酶激活受体)-4 拮抗剂和 Xa 因子抑制剂联合应用的抗血栓作用

Mohammed N Meah, Jennifer Raftis, Simon J Wilson, Vidya Perera, Samira M Garonzik, Bindu Murthy, J Gerry Everlof, Ronald Aronson, Joseph Luettgen, David E Newby

Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors

临床候选药物BMS-906024的发现:一种用于治疗白血病和实体瘤的强效泛Notch抑制剂

Gavai, Ashvinikumar V; Quesnelle, Claude; Norris, Derek; Han, Wen-Ching; Gill, Patrice; Shan, Weifang; Balog, Aaron; Chen, Ke; Tebben, Andrew; Rampulla, Richard; Wu, Dauh-Rurng; Zhang, Yingru; Mathur, Arvind; White, Ronald; Rose, Anne; Wang, Haiqing; Yang, Zheng; Ranasinghe, Asoka; D'Arienzo, Celia; Guarino, Victor; Xiao, Lan; Su, Ching; Everlof, Gerry; Arora, Vinod; Shen, Ding Ren; Cvijic, Mary Ellen; Menard, Krista; Wen, Mei-Li; Meredith, Jere; Trainor, George; Lombardo, Louis J; Olson, Richard; Baran, Phil S; Hunt, John T; Vite, Gregory D; Fischer, Bruce S; Westhouse, Richard A; Lee, Francis Y