日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tumor microenvironment-activated ferritin nanovector enables enhanced tumor delivery of KRAS(G12C) inhibitors and degraders

肿瘤微环境激活的铁蛋白纳米载体可增强KRAS(G12C)抑制剂和降解剂的肿瘤递送。

Abbinantefina, Annalisa Pia; Tito, Claudia; Masciarelli, Silvia; Tisci, Giada; Sortoluzzi, Siria; Ceci, Pierpaolo; Falvo, Elisabetta; Exertier, Cécile; Troilo, Francesca; Petrozza, Vincenzo; Mai, Antonello; Rotili, Dante; Fazi, Francesco; Colotti, Gianni

Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis

片段合并、生长和连接可鉴定用于治疗利什曼病的新型锥虫硫酮还原酶抑制剂

Cécile Exertier, Alessandra Salerno, Lorenzo Antonelli, Annarita Fiorillo, Riccardo Ocello, Francesca Seghetti, Jessica Caciolla, Elisa Uliassi, Matteo Masetti, Eleonora Fiorentino, Stefania Orsini, Trentina Di Muccio, Andrea Ilari, Maria Laura Bolognesi

Sorcin in Cancer Development and Chemotherapeutic Drug Resistance

索辛在癌症发展和化疗耐药性中的作用

Exertier, Cécile; Antonelli, Lorenzo; Fiorillo, Annarita; Bernardini, Roberta; Colotti, Beatrice; Ilari, Andrea; Colotti, Gianni

Structural insights into the DNA recognition mechanism by the bacterial transcription factor PdxR

细菌转录因子 PdxR 对 DNA 识别机制的结构解析

Freda, Ida; Exertier, Cécile; Barile, Anna; Chaves-Sanjuan, Antonio; Vega, Mirella Vivoli; Isupov, Michail N; Harmer, Nicholas J; Gugole, Elena; Swuec, Paolo; Bolognesi, Martino; Scipioni, Anita; Savino, Carmelinda; Di Salvo, Martino Luigi; Contestabile, Roberto; Vallone, Beatrice; Tramonti, Angela; Montemiglio, Linda Celeste

Innovative Approach for a Classic Target: Fragment Screening on Trypanothione Reductase Reveals New Opportunities for Drug Design

针对经典靶点的创新方法:锥虫硫还原酶片段筛选揭示药物设计的新机遇

Fiorillo, Annarita; Colotti, Gianni; Exertier, Cécile; Liuzzi, Anastasia; Seghetti, Francesca; Salerno, Alessandra; Caciolla, Jessica; Ilari, Andrea

Probing the Role of Murine Neuroglobin CDloop-D-Helix Unit in CO Ligand Binding and Structural Dynamics

探究小鼠神经球蛋白CD环-D螺旋单元在CO配体结合和结构动力学中的作用

Exertier, Cécile; Sebastiani, Federico; Freda, Ida; Gugole, Elena; Cerutti, Gabriele; Parisi, Giacomo; Montemiglio, Linda Celeste; Becucci, Maurizio; Viappiani, Cristiano; Bruno, Stefano; Savino, Carmelinda; Zamparelli, Carlotta; Anselmi, Massimiliano; Abbruzzetti, Stefania; Smulevich, Giulietta; Vallone, Beatrice

ALS2-Related Motor Neuron Diseases: From Symptoms to Molecules

ALS2相关运动神经元疾病:从症状到分子机制

Miceli, Marcello; Exertier, Cécile; Cavaglià, Marco; Gugole, Elena; Boccardo, Marta; Casaluci, Rossana Rita; Ceccarelli, Noemi; De Maio, Alessandra; Vallone, Beatrice; Deriu, Marco A

Crystal structure and functional characterization of an oligosaccharide dehydrogenase from Pycnoporus cinnabarinus provides insights into fungal breakdown of lignocellulose

对朱砂大孔菌(Pycnoporus cinnabarinus)寡糖脱氢酶的晶体结构和功能表征,揭示了真菌分解木质纤维素的机制。

Cerutti, Gabriele; Gugole, Elena; Montemiglio, Linda Celeste; Turbé-Doan, Annick; Chena, Dehbia; Navarro, David; Lomascolo, Anne; Piumi, François; Exertier, Cécile; Freda, Ida; Vallone, Beatrice; Record, Eric; Savino, Carmelinda; Sciara, Giuliano

The Nuts and Bolts of SARS-CoV-2 Spike Receptor-Binding Domain Heterologous Expression

SARS-CoV-2 刺突受体结合域异源表达的具体细节

Mariano Maffei, Linda Celeste Montemiglio, Grazia Vitagliano, Luigi Fedele, Shaila Sellathurai, Federica Bucci, Mirco Compagnone, Valerio Chiarini, Cécile Exertier, Alessia Muzi, Giuseppe Roscilli, Beatrice Vallone, Emanuele Marra

Ligand pathways in neuroglobin revealed by low-temperature photodissociation and docking experiments

低温光解离和对接实验揭示神经球蛋白中的配体通路

Ardiccioni, Chiara; Arcovito, Alessandro; Della Longa, Stefano; van der Linden, Peter; Bourgeois, Dominique; Weik, Martin; Montemiglio, Linda Celeste; Savino, Carmelinda; Avella, Giovanna; Exertier, Cécile; Carpentier, Philippe; Prangé, Thierry; Brunori, Maurizio; Colloc'h, Nathalie; Vallone, Beatrice