日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inducing TRIB2-targeted protein degradation to reverse chemoresistance in acute myeloid leukaemia

诱导 TRIB2 靶向蛋白降解以逆转急性髓系白血病的化疗耐药性

Rigby, Evie; Fasanella Masci, Francesca; Narayanan, Akshara; Kania, Elzbieta; Harris, John A; Williams, Jamie; Zhang, Binghua; Liu, Lijun; Richmond, Laura; Zhou, Fengtao; Ding, Ke; Carmody, Ruaidhrí J; Eyers, Patrick A; Keeshan, Karen

RAF inhibitors activate the integrated stress response by direct activation of GCN2

RAF抑制剂通过直接激活GCN2来激活整合应激反应。

Gilley, Rebecca; Kidger, Andrew M; Neill, Graham; Morrison, Eve; Severson, Paul; Byrne, Dominic P; Kenneth, Niall S; Bollag, Gideon; Zhang, Chao; Maia de Oliveira, Taiana; Eyers, Patrick A; Bayliss, Richard; Masson, Glenn R; Cook, Simon J

PSKH1 kinase activity is differentially modulated via allosteric binding of Ca(2+) sensor proteins

PSKH1激酶活性受Ca(2+)传感器蛋白变构结合的差异性调节。

Horne, Christopher R; Dite, Toby A; Young, Samuel N; Mather, Lucy J; Dagley, Laura F; Johnson, Jared L; Yaron-Barir, Tomer M; Huntsman, Emily M; Daly, Leonard A; Byrne, Dominic P; Cadell, Antonia L; Ng, Boaz H; Yousef, Jumana; Multari, Dylan H; Shen, Lianju; McAloon, Luke M; Manning, Gerard; Febbraio, Mark A; Means, Anthony R; Cantley, Lewis C; Tanzer, Maria C; Croucher, David R; Eyers, Claire E; Eyers, Patrick A; Scott, John W; Murphy, James M

Redox regulation and dynamic control of brain-selective kinases BRSK1/2 in the AMPK family through cysteine-based mechanisms.

通过半胱氨酸机制对 AMPK 家族中脑选择性激酶 BRSK1/2 进行氧化还原调节和动态控制

Bendzunas George N, Byrne Dominic P, Shrestha Safal, Daly Leonard A, Oswald Sally O, Katiyar Samiksha, Venkat Aarya, Yeung Wayland, Eyers Claire E, Eyers Patrick A, Kannan Natarajan

Autophagy inhibitors block pathogenic NET release in immune-mediated inflammatory disease without impairing host defence.

自噬抑制剂可阻断免疫介导的炎症疾病中致病性 NET 的释放,而不会损害宿主的防御能力。

Nolan Andy, Foulkes Daniel M, Fairweather Emma E, Alarcon Michele Fresneda, Linford Christina, Sellin Andrew, McLaren Zoe, Eyers Patrick A, Wright Helen L

Structural and evolutionary insights into understudied bacterial serine-threonine pseudokinase families

对研究不足的细菌丝氨酸/苏氨酸假激酶家族的结构和进化见解

O'Boyle, Brady; Bhowmik, Debarshi Ryan; Eyers, Patrick A; Byrne, Dominic P; Kannan, Natarajan

Applying a Conservation-Based Approach for Predicting Novel Phosphorylation Sites in Eukaryotes and Evaluating Their Functional Relevance

应用基于保守性的方法预测真核生物中新的磷酸化位点并评估其功能相关性

Kalyuzhnyy, Anton; Eyers, Patrick A; Eyers, Claire E; Deutsch, Eric W; Jones, Andrew R

Redox Regulation of Brain Selective Kinases BRSK1/2: Implications for Dynamic Control of the Eukaryotic AMPK family through Cys-based mechanisms

脑选择性激酶 BRSK1/2 的氧化还原调节:通过基于 Cys 的机制对真核 AMPK 家族进行动态控制的意义

George N Bendzunas, Dominic P Byrne, Safal Shrestha, Leonard A Daly, Sally O Oswald, Samiksha Katiyar, Aarya Venkat, Wayland Yeung, Claire E Eyers, Patrick A Eyers, Natarajan Kannan

Profiling the Human Phosphoproteome to Estimate the True Extent of Protein Phosphorylation

通过分析人类磷酸化蛋白质组来估计蛋白质磷酸化的真实程度

Kalyuzhnyy, Anton; Eyers, Patrick A; Eyers, Claire E; Bowler-Barnett, Emily; Martin, Maria J; Sun, Zhi; Deutsch, Eric W; Jones, Andrew R

Exploring the Conformational Landscape and Stability of Aurora A Using Ion-Mobility Mass Spectrometry and Molecular Modeling.

利用离子迁移质谱和分子建模探索 Aurora A 的构象景观和稳定性

Tomlinson Lauren J, Batchelor Matthew, Sarsby Joscelyn, Byrne Dominic P, Brownridge Philip J, Bayliss Richard, Eyers Patrick A, Eyers Claire E