日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Activation and inhibition of sirtuins: From bench to bedside

sirtuins 的激活和抑制:从实验室到临床

Fiorentino, Francesco; Fabbrizi, Emanuele; Mai, Antonello; Rotili, Dante

An Amazing 30-Year Journey around the DABO Family: A Medicinal Chemistry Lesson on a Versatile Class of Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

DABO家族30年奇妙历程:一堂关于多功能非核苷类HIV-1逆转录酶抑制剂的药物化学课

Fabbrizi, Emanuele; Chernyshov, Vladimir V; Fiorentino, Francesco; Sbardella, Gianluca; Ragno, Rino; Nawrozkij, Maxim; Ivanov, Roman; Rotili, Dante; Mai, Antonello

Duplexed CeTEAM drug biosensors reveal determinants of PARP inhibitor selectivity in cells.

双链CeTEAM药物生物传感器揭示了细胞中PARP抑制剂选择性的决定因素

Pires Maria J, Alam Seher, Lovric Alen, Fabbrizi Emanuele, Rotili Dante, Altun Mikael, Valerie Nicholas C K

Tranylcypromine-Based LSD1 Inhibitors as Useful Agents to Reduce Viability of Schistosoma mansoni

基于反式环丙胺的LSD1抑制剂可有效降低曼氏血吸虫的存活率

Fabbrizi, Emanuele; Hailu, Gebremedhin Solomon; Ganesan, A; Fioravanti, Rossella; Zwergel, Clemens; Lambona, Chiara; Valente, Sergio; Fianco, Giulia; Iuzzolino, Angela; Trisciuoglio, Daniela; Caroli, Jonatan; Mattevi, Andrea; Häberli, Cécile; Keiser, Jennifer; Rotili, Dante; Mai, Antonello

Benzodeazaoxaflavin Sirtuin Inhibitors Inhibit Schistosoma mansoni Sirt2 and Cause Phenotypic Changes and Lethality in Schistosomula and Adult Worm Stages.

苯并二氮杂黄素 Sirtuin 抑制剂抑制曼氏血吸虫 Sirt2,导致血吸虫幼虫和成虫阶段的表型变化和致死性。

Gimmelli Roberto, Papoff Giuliana, Fabbrizi Emanuele, Guida Michela, Lalli Cristiana, Saccoccia Fulvio, Häberli Cécile, Keiser Jennifer, Monaldi Daria, Jung Manfred, Romier Christophe, Rotili Dante, Mai Antonello, Ruberti Giovina

Development of C646-Based Proteolysis Targeting Chimeras Degraders of the Lysine Acetyltransferases CBP and p300

基于C646的蛋白水解靶向嵌合体降解赖氨酸乙酰转移酶CBP和p300的开发

Fiorentino, Francesco; Spriano, Filippo; Tomaselli, Daniela; Risi, Giorgia; Fabbrizi, Emanuele; Pecci, Valeria; Nanni, Simona; Bertoni, Francesco; Rotili, Dante; Mai, Antonello

Transmission-Blocking Strategies for Malaria Eradication: Recent Advances in Small-Molecule Drug Development

疟疾根除的传播阻断策略:小分子药物研发的最新进展

Appetecchia, Federico; Fabbrizi, Emanuele; Fiorentino, Francesco; Consalvi, Sara; Biava, Mariangela; Poce, Giovanna; Rotili, Dante

Emerging Roles of SIRT5 in Metabolism, Cancer, and SARS-CoV-2 Infection

SIRT5在代谢、癌症和SARS-CoV-2感染中的新兴作用

Fabbrizi, Emanuele; Fiorentino, Francesco; Carafa, Vincenzo; Altucci, Lucia; Mai, Antonello; Rotili, Dante