Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation
设计新型二取代咪唑并[1,2-b]哒嗪衍生物作为选择性Haspin抑制剂。合成、结合模式及抗癌生物学评价
期刊:Journal of Enzyme Inhibition and Medicinal Chemistry
影响因子:5.4
doi:10.1080/14756366.2020.1825408
Elie, Jonathan; Feizbakhsh, Omid; Desban, Nathalie; Josselin, Béatrice; Baratte, Blandine; Bescond, Amandine; Duez, Julien; Fant, Xavier; Bach, Stéphane; Marie, Dominique; Place, Matthieu; Ben Salah, Sami; Chartier, Agnes; Berteina-Raboin, Sabine; Chaikuad, Apirat; Knapp, Stefan; Carles, Fabrice; Bonnet, Pascal; Buron, Frédéric; Routier, Sylvain; Ruchaud, Sandrine