日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Comparative metabolism of conjugated and unconjugated pterins in Crithidia, Leishmania and African trypanosomes

锥虫、利什曼原虫和非洲锥虫中结合型和非结合型蝶呤的代谢比较

Ong, Han B; Wyllie, Susan; Fairlamb, Alan H

Validation of Trypanosoma cruzi inactivation techniques for laboratory use

实验室用克氏锥虫灭活技术的验证

MacLean, Lorna M; Ariyanayagam, Mark; Sastry, Lalitha; Paterson, Christy; De Rycker, Manu; Fairlamb, Alan H

The critical role of mode of action studies in kinetoplastid drug discovery

作用机制研究在动质体药物发现中的关键作用

Fairlamb, Alan H; Wyllie, Susan

Surmounting structural barriers to tackle endemic infectious diseases

克服结构性障碍以应对地方性传染病

Calderón, Felix; Fairlamb, Alan H; Strange, Mike; Williams, Pauline; Nathan, Carl F

New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruzi

一种新型 8-硝基喹啉酮衍生物对布氏锥虫和克氏锥虫均表现出亚微摩尔级的体外活性。

Pedron, Julien; Boudot, Clotilde; Brossas, Jean-Yves; Pinault, Emilie; Bourgeade-Delmas, Sandra; Sournia-Saquet, Alix; Boutet-Robinet, Elisa; Destere, Alexandre; Tronnet, Antoine; Bergé, Justine; Bonduelle, Colin; Deraeve, Céline; Pratviel, Geneviève; Stigliani, Jean-Luc; Paris, Luc; Mazier, Dominique; Corvaisier, Sophie; Since, Marc; Malzert-Fréon, Aurélie; Wyllie, Susan; Milne, Rachel; Fairlamb, Alan H; Valentin, Alexis; Courtioux, Bertrand; Verhaeghe, Pierre

The Q(i) Site of Cytochrome b is a Promiscuous Drug Target in Trypanosoma cruzi and Leishmania donovani

细胞色素b的Q(i)位点是克氏锥虫和杜氏利什曼原虫的多种药物靶点之一。

Wall, Richard J; Carvalho, Sandra; Milne, Rachel; Bueren-Calabuig, Juan A; Moniz, Sonia; Cantizani-Perez, Juan; MacLean, Lorna; Kessler, Albane; Cotillo, Ignacio; Sastry, Lalitha; Manthri, Sujatha; Patterson, Stephen; Zuccotto, Fabio; Thompson, Stephen; Martin, Julio; Marco, Maria; Miles, Timothy J; De Rycker, Manu; Thomas, Michael G; Fairlamb, Alan H; Gilbert, Ian H; Wyllie, Susan

Nongenotoxic 3-Nitroimidazo[1,2-a]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial Activity

非基因毒性的3-硝基咪唑并[1,2-a]吡啶类化合物是NTR1的底物,在体外显示出强大的抗利什曼原虫活性。

Fersing, Cyril; Basmaciyan, Louise; Boudot, Clotilde; Pedron, Julien; Hutter, Sébastien; Cohen, Anita; Castera-Ducros, Caroline; Primas, Nicolas; Laget, Michèle; Casanova, Magali; Bourgeade-Delmas, Sandra; Piednoel, Mélanie; Sournia-Saquet, Alix; Belle Mbou, Valère; Courtioux, Bertrand; Boutet-Robinet, Élisa; Since, Marc; Milne, Rachel; Wyllie, Susan; Fairlamb, Alan H; Valentin, Alexis; Rathelot, Pascal; Verhaeghe, Pierre; Vanelle, Patrice; Azas, Nadine

Substituted Aminoacetamides as Novel Leads for Malaria Treatment

取代氨基乙酰胺作为疟疾治疗的新型先导化合物

Norcross, Neil R; Wilson, Caroline; Baragaña, Beatriz; Hallyburton, Irene; Osuna-Cabello, Maria; Norval, Suzanne; Riley, Jennifer; Fletcher, Daniel; Sinden, Robert; Delves, Michael; Ruecker, Andrea; Duffy, Sandra; Meister, Stephan; Antonova-Koch, Yevgeniya; Crespo, Benigno; de Cózar, Cristina; Sanz, Laura M; Gamo, Francisco Javier; Avery, Vicky M; Frearson, Julie A; Gray, David W; Fairlamb, Alan H; Winzeler, Elizabeth A; Waterson, David; Campbell, Simon F; Willis, Paul A; Read, Kevin D; Gilbert, Ian H

Cyclin-dependent kinase 12 is a drug target for visceral leishmaniasis

细胞周期蛋白依赖性激酶12是内脏利什曼病的一种药物靶点。

Wyllie, Susan; Thomas, Michael; Patterson, Stephen; Crouch, Sabrinia; De Rycker, Manu; Lowe, Rhiannon; Gresham, Stephanie; Urbaniak, Michael D; Otto, Thomas D; Stojanovski, Laste; Simeons, Frederick R C; Manthri, Sujatha; MacLean, Lorna M; Zuccotto, Fabio; Homeyer, Nadine; Pflaumer, Hannah; Boesche, Markus; Sastry, Lalitha; Connolly, Paul; Albrecht, Sebastian; Berriman, Matt; Drewes, Gerard; Gray, David W; Ghidelli-Disse, Sonja; Dixon, Susan; Fiandor, Jose M; Wyatt, Paul G; Ferguson, Michael A J; Fairlamb, Alan H; Miles, Timothy J; Read, Kevin D; Gilbert, Ian H

Antitrypanosomal 8-Hydroxy-Naphthyridines Are Chelators of Divalent Transition Metals

抗锥虫8-羟基萘啶类化合物是二价过渡金属螯合剂

Wall, Richard J; Moniz, Sonia; Thomas, Michael G; Norval, Suzanne; Ko, Eun-Jung; Marco, Maria; Miles, Timothy J; Gilbert, Ian H; Horn, David; Fairlamb, Alan H; Wyllie, Susan