日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

2-Arylbenzofurans as Selective Cholinesterase Inhibitors: Design, Synthesis, and Evaluation as Alzheimer's Disease Agents

2-芳基苯并呋喃类化合物作为选择性胆碱酯酶抑制剂:设计、合成及作为阿尔茨海默病治疗药物的评价

Delogu, Giovanna Lucia; Begala, Michela; Novás, Manuel; Matos, Maria João; Piras, Franca; Floris, Sonia; Pintus, Francesca; Mancinelli, Michele; Era, Benedetta; Fais, Antonella

Valorization of Pistacia lentiscus L. Hydrodistillation By-Products: Phytochemical Profile and Multitarget Anti-Aging Activity of an Aqueous Extract

乳香黄连木水蒸馏副产物的增值利用:水提取物的植物化学成分分析及多靶点抗衰老活性

Fais, Antonella; Pintus, Francesca; Era, Benedetta; Floris, Sonia; Urru, Giulia; Sanjust, Enrico; Cocco, Emma; Maxia, Andrea; Masala, Valentina; Tuberoso, Carlo Ignazio Giovanni

Investigating the Ligand-Binding Properties of N-arylbenzimidazoles as Novel Elastase Inhibitors

研究N-芳基苯并咪唑类化合物作为新型弹性蛋白酶抑制剂的配体结合特性

Pitasi, Giovanna; Floris, Sonia; Mancuso, Francesca; Savoca, Giulia; Gitto, Rosaria; Fais, Antonella; De Luca, Laura

The Anti-Angiogenic Effect of Cynara cardunculus L. subsp. cardunculus Waste Product

蓟菜(Cynara cardunculus L. subsp. cardunculus)废弃物的抗血管生成作用

Cacciola, Anna; D'Angelo, Valeria; De Gaetano, Federica; Fais, Antonella; Germanò, Maria Paola; Masala, Valentina; Olla, Stefania; Pistarà, Venerando; Stancanelli, Rosanna; Tuberoso, Carlo Ignazio Giovanni; Ventura, Cinzia Anna

Sustainable Synthesis of 1,2-Disubstituted Benzimidazoles as Promising α-Glucosidase Inhibitors: In Vitro and In Silico Evaluation

1,2-二取代苯并咪唑类化合物作为有前景的α-葡萄糖苷酶抑制剂的可持续合成:体外和计算机模拟评价

Tocco, Graziella; Laus, Antonio; Manis, Cristina; Caboni, Pierluigi; Fais, Antonella; Era, Benedetta

Xanthine Oxidase-Dependent Activation of NLPR3 Inflammasome in Epithelial Cells Sustains Inflammation in Inflammatory Bowel Disease

黄嘌呤氧化酶依赖性NLPR3炎症小体在肠上皮细胞中的激活维持炎症

Di Petrillo, Amalia; Fais, Antonella; Raho, Nicola; Era, Benedetta; Cannea, Faustina Barbara; Padiglia, Alessandra; Grecu, Eleonora; Murtas, Daniela; Maxia, Cristina; Sogos, Valeria; Porcedda, Clara; Caboni, Pierluigi; Demurtas, Mauro; Favale, Agnese; Onali, Sara; Fantini, Massimo Claudio

Inhibition of α-Glucosidase Activity and Islet Amyloid PolyPeptide Fibril Formation by Rubusulmifolius Fruit Extract: A Potential Therapeutic Approach for Type 2 Diabetes Mellitus

覆盆子果实提取物对α-葡萄糖苷酶活性和胰岛淀粉样多肽原纤维形成的抑制作用:一种治疗2型糖尿病的潜在方法

Floris, Sonia; Noli, Barbara; Cocco, Cristina; Fais, Antonella; Era, Benedetta; Tuberoso, Carlo Ignazio Giovanni; Masala, Valentina; Piras, Franca; Sogos, Valeria; Di Petrillo, Amalia; De Agostini, Antonio; Pintus, Francesca; Sanna, Cinzia

Structure-based design and evaluation of tyrosinase inhibitors targeting both human and mushroom isozymes.

基于结构的酪氨酸酶抑制剂的设计和评价,靶向人类和蘑菇同工酶

Mirabile Salvatore, Pitasi Giovanna, Floris Sonia, Schira Kristina, Khettabi Lyna, Soler-Lopez Montserrat, Scheuermann Jörg, Gitto Rosaria, Germanò Maria Paola, Fais Antonella, De Luca Laura

Computational Approach to Identifying New Chemical Entities as Elastase Inhibitors with Potential Antiaging Effects

利用计算方法识别具有潜在抗衰老作用的新型弹性蛋白酶抑制剂。

Pitasi, Giovanna; Brancale, Andrea; Floris, Sonia; Fais, Antonella; Gitto, Rosaria; De Luca, Laura

Biological Potential of Asphodelus microcarpus Extracts: α-Glucosidase and Antibiofilm Activities In Vitro

小果芦荟提取物的生物学潜力:体外α-葡萄糖苷酶和抗生物膜活性

Floris, Sonia; Pintus, Francesca; Fais, Antonella; Era, Benedetta; Raho, Nicola; Siguri, Chiara; Orrù, Germano; Fais, Sara; Tuberoso, Carlo Ignazio Giovanni; Olla, Stefania; Di Petrillo, Amalia