日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design of a Targeted Covalent Probe to Interrogate the DNA Polymerase Activity of Polθ

设计靶向共价探针以检测Polθ的DNA聚合酶活性

Bubenik, Monica; Mader, Pavel; Orlicky, Stephen; Perryman, Alexander L; Hamel, Martine; Godbout, Claude; Falgueyret, Jean-Pierre; Kurinov, Igor; Wong, Cassandra; Gingras, Anne Claude; Mamane, Yael; Zinda, Michael; Morris, Stephen J; Gallant, Michel; Sfeir, Agnel; Black, W Cameron; Durocher, Daniel; Zimmermann, Michal; Sicheri, Frank

In vitro characterization of MK-1439, a novel HIV-1 nonnucleoside reverse transcriptase inhibitor.

体外表征新型 HIV-1 非核苷类逆转录酶抑制剂 MK-1439

Lai Ming-Tain, Feng Meizhen, Falgueyret Jean-Pierre, Tawa Paul, Witmer Marc, DiStefano Daniel, Li Yuan, Burch Jason, Sachs Nancy, Lu Meiqing, Cauchon Elizabeth, Campeau Louis-Charles, Grobler Jay, Yan Youwei, Ducharme Yves, Côté Bernard, Asante-Appiah Ernest, Hazuda Daria J, Miller Michael D

Automethylation of protein arginine methyltransferase 6 (PRMT6) regulates its stability and its anti-HIV-1 activity

蛋白质精氨酸甲基转移酶6 (PRMT6) 的自身甲基化调节其稳定性及其抗HIV-1活性。

Singhroy, Diane N; Mesplède, Thibault; Sabbah, Arielle; Quashie, Peter K; Falgueyret, Jean-Pierre; Wainberg, Mark A