日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a novel AhR-CYP1A1 axis activator for mitigating inflammatory diseases using an in situ functional imaging assay

利用原位功能成像分析法发现了一种新型AhR-CYP1A1轴激活剂,可用于缓解炎症性疾病。

Zhang, Feng; Zhao, Bei; Fan, Yufan; Qin, Lanhui; Shi, Jinhui; Chen, Lin; Xu, Leizhi; Jin, Xudong; Sun, Mengru; Deng, Hongping; Zeng, Hairong; Xiao, Zhangping; Yang, Xin; Ge, Guangbo

Discovery of novel butyrylcholinesterase inhibitors for treating Alzheimer's disease

发现用于治疗阿尔茨海默病的新型丁酰胆碱酯酶抑制剂

Sang, Zhipei; Huang, Shuheng; Tan, Wanying; Ban, Yujuan; Wang, Keren; Fan, Yufan; Chen, Hongsong; Zhang, Qiyao; Liang, Chanchan; Mi, Jing; Gao, Yunqi; Zhang, Ya; Liu, Wenmin; Wang, Jianta; Dong, Wu; Tan, Zhenghuai; Tang, Lei; Luo, Haibin

Discovery of orally active and serine-targeting covalent inhibitors against hCES2A for ameliorating irinotecan-triggered gut toxicity

发现口服有效的、靶向丝氨酸的hCES2A共价抑制剂,以改善伊立替康引发的肠道毒性

Zhang, Ya; Fan, Yufan; Song, Yunqing; Zhu, Guanghao; Li, Xinjuan; Huang, Jian; Guo, Xinrui; Luan, Changhai; Kang, Dongning; Chen, Lu; Xiao, Zhangping; Guo, Zhaobin; Zeng, Hairong; Chen, Dapeng; Sang, Zhipei; Ge, Guangbo

High-efficient discovering the potent anti-Notum agents from herbal medicines for combating glucocorticoid-induced osteoporosis.

高效发现草药中强效抗骨质疏松剂,用于对抗糖皮质激素引起的骨质疏松症

Song Yuqing, Zhang Feng, Guo Jia, Fan Yufan, Zeng Hairong, Sun Mengru, Qian Jun, Qi Shenglan, Chen Zihan, Jin Xudong, Song Yunqing, Tian Tian, Qian Zhi, Sun Yao, Tian Zhenhao, Yu Baoqing, Ge Guangbo

Functional Imaging of CYP3A4 at Multiple Dimensions Using an AI-Driven High Performance Fluorogenic Substrate

利用人工智能驱动的高性能荧光底物对CYP3A4进行多维度功能成像

Zhang, Feng; Song, Lilin; Wang, Ruixuan; Zhao, Bei; Huang, Jian; Wu, Luling; Fan, Yufan; Lin, Hong; Jiang, Zhengtao; Yang, Xiaodi; Zeng, Hairong; Yang, Xin; James, Tony D; Ge, Guangbo

An optimized CYP3A4-activatable fluorogenic sensor for in situ functional imaging and multi-dimensional inhibitor assessment

一种优化的CYP3A4激活型荧光传感器,用于原位功能成像和多维抑制剂评估

Zhang, Feng; Fan, Yufan; Luo, Mei; Huang, Jian; Zhao, Bei; Chen, Lin; Zhu, Guanghao; Xiong, Yuan; Lin, Hong; Xu, Chuting; Yang, Xiaodi; James, Tony D; Ge, Guangbo

A Novel Fluorescence-Based Microplate Assay for High-Throughput Screening of hSULT1As Inhibitors

一种用于高通量筛选hSULT1As抑制剂的新型基于荧光的微孔板检测方法

Niu, Xiaoting; Fan, Yufan; Zou, Liwei; Ge, Guangbo

FABP4 in macrophages facilitates obesity-associated pancreatic cancer progression via the NLRP3/IL-1β axis

巨噬细胞中的 FABP4 通过 NLRP3/IL-1β 轴促进肥胖相关的胰腺癌进展

Jian Yang, Shujie Liu, Yongzheng Li, Zhiyao Fan, Yufan Meng, Bin Zhou, Guangyong Zhang, Hanxiang Zhan

[Advances in chromatography in the study of drug-plasma protein interactions]

[色谱技术在药物-血浆蛋白相互作用研究中的进展]

Bai, Yu; Fan, Yufan; Ge, Guangbo; Wang, Fangjun