日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Human Mass Balance and Metabolism Study of [(14)C]-Ubrogepant in Healthy Male Adults

一项关于[(14)C]-Ubrogepant在健康成年男性中的人体质量平衡和代谢研究

Boinpally, Ramesh R; Rowe, Joshua; Chandrasekar, Pushpa; White, Rebecca B; Marcantonio, Eugene E; Trainor, Nicole; Liang, Yuexia; Maciolek, Cheri; Small, James H; Houle, Robert; Hafey, Michael J; Xie, Huizhi; Yabut, Jocelyn; Fandozzi, Christine

2025 White Paper on Recent Issues in Bioanalysis: What is the Future of Bioanalytical LIMS? AI/ML Integration in Bioanalysis; Tear Sample Collection; Radiolabeled Mass Balance Studies; Chiral Assays; Bioanalysis of Antibody-Oligonucleotide & Bicycle Drug Conjugates (PART 1A - Recommendations on Mass Spectrometry Assays, Chromatography, Sample Preparation and Regulated Bioanalysis Sampling, Validating, Analyzing & Reporting PART 1B - Regulatory Agencies' Input on Regulated Bioanalysis/BMV)

2025 年生物分析最新问题白皮书:生物分析 LIMS 的未来是什么?人工智能/机器学习在生物分析中的应用;泪液样本采集;放射性标记质量平衡研究;手性分析;抗体-寡核苷酸和环状药物偶联物的生物分析(第一部分 A - 关于质谱分析、色谱、样品制备和受监管生物分析采样、验证、分析和报告的建议;第一部分 B - 监管机构对受监管生物分析/生物质量监测的意见)

Wojcik, John; Qian, Mark; Rosenbaum, Anton I; Maes, Estelle; Xue, Yongjun; Kochansky, Christopher; Boer, Jason; Chen, Linzhi; Descloux, Sandrine; Garofolo, Fabio; Johnson, Jay; Kaur, Surinder; Lassman, Michael; McGregor, Jessica; O'Callaghan, Lisa; Sikorski, Timothy; Wan, Katty; Wang, Shunhai; Zheng, Naiyu; Zhang, Guodong; Hoover, Michael; Wang, Jian; Yuan, Long; Ji, Qin; Jones, Barry; Boyanapalli, Ramakrishna; Chen, Jian; Dobson, Christine; Dong, Linlin; Ferrari, Luca; Fu, Yunlin; Gong, Chao; Ivanova, Dany; Li, Jing; Licea-Perez, Hermes; Liu, Aihua; Tang, Xiaonan; Tao, Lin; Tweed, Joseph; Eddy, John; Francis, Jennifer; Kavetska, Olga; Araya, Marcela; Foley, Timothy; Andisik, Matthew; Belfast, Mary; Borbridge, Lisa; Cho, Seongeun Julia; Colligan, Liliana; Dasgupta, Arindam; Edmison, Anna; Fandozzi, Christine; Galliccia, Fabrizio; Kim, Yeoun Jin; Lu, Yang; Massip, Anne-Marie; Shakleya, Diaa; Tampal, Nilufer; Neto, Joao Tavares; Thomas, Justina; Wang, Jin; Wang, Linna; Wang, Ying; Whale, Emma; Wiberg, Megan; Yang, Li

Aeromonas nosocomial cluster: Investigation review of possible modes of transmission

气单胞菌院内感染群:对可能传播途径的调查回顾

Wan, Yuxi; Chen, Qiangguo; Yan, Tingting; Liu, Ching-Hsuan; Lin, Yuan-Yu; Pellerino, A; Marchesani, E; Bertero, L; Ricci, A; Mangherini, L; Bruno, F; Soffietti, R; Rudà, R; Riviere-Cazaux, C; Mo, W; Dong, X; Luo, S; Wang, A; Du, P; Ghadimi, K; Warrington, A; Burns, T; Messman, Riley D; Swanson, Rebecca M; Lemley, Caleb O; Fandozzi, Eva; Smith, Caroline; Megli, Christina; Williams, Monray E; Thomas, Clayton; Grantham, James; Lute, Emily; Davidson, Jerod; Cowden, Scott; Nutt, Jamie; Bisht, Anjali; Gray, Hannah; Caldera, JR; Yang, Shangxin; Uslan, Dan

Pharmacokinetic Interactions between the Hepatitis C Virus Inhibitors Elbasvir and Grazoprevir and HIV Protease Inhibitors Ritonavir, Atazanavir, Lopinavir, and Darunavir in Healthy Volunteers

在健康志愿者中,丙型肝炎病毒抑制剂艾尔巴韦和格拉佐普韦与HIV蛋白酶抑制剂利托那韦、阿扎那韦、洛匹那韦和达芦那韦之间的药代动力学相互作用

Feng, Hwa-Ping; Caro, Luzelena; Fandozzi, Christine; Chu, Xiaoyan; Guo, Zifang; Talaty, Jennifer; Panebianco, Deborah; Dunnington, Katherine; Du, Lihong; Hanley, William D; Fraser, Iain P; Mitselos, Anna; Denef, Jean-Francois; De Lepeleire, Inge; de Hoon, Jan N; Vandermeulen, Corinne; Marshall, William L; Jumes, Patricia; Huang, Xiaobi; Martinho, Monika; Valesky, Robert; Butterton, Joan R; Iwamoto, Marian; Yeh, Wendy W

Effect of Hepatic Impairment on the Pharmacokinetics of Grazoprevir, a Hepatitis C Virus Protease Inhibitor

肝功能损害对丙型肝炎病毒蛋白酶抑制剂格拉瑞韦药代动力学的影响

Caro, Luzelena; Wenning, Larissa; Guo, Zifang; Fraser, Iain P; Fandozzi, Christine; Talaty, Jennifer; Panebianco, Deborah; Ho, Maureen; Uemura, Naoto; Reitmann, Christina; Angus, Peter; Gane, Edward; Marbury, Thomas; Smith, William B; Iwamoto, Marian; Butterton, Joan R; Yeh, Wendy W

MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants

MK-5172,一种选择性抑制丙型肝炎病毒NS3/4a蛋白酶的药物,对多种基因型和耐药变异株均具有广泛活性。

Draper, Michael P; Weir, S; Macone, A; Donatelli, J; Trieber, C A; Tanaka, S K; Levy, Stuart B; P, Shahul Hameed; Solapure, Suresh; Mukherjee, Kakoli; Nandi, Vrinda; Waterson, David; Shandil, Radha; Balganesh, Meenakshi; Sambandamurthy, Vasan K; Raichurkar, Anand Kumar; Deshpande, Abhijeet; Ghosh, Anirban; Awasthy, Disha; Shanbhag, Gajanan; Sheikh, Gulebahar; McMiken, Helen; Puttur, Jayashree; Reddy, Jitendar; Werngren, Jim; Read, Jon; Kumar, Mahesh; R, Manjunatha; Chinnapattu, Murugan; Madhavapeddi, Prashanti; Manjrekar, Praveena; Basu, Reetobrata; Gaonkar, Sheshagiri; Sharma, Sreevalli; Hoffner, Sven; Humnabadkar, Vaishali; Subbulakshmi, Venkita; Panduga, Vijender; Summa, Vincenzo; Ludmerer, Steven W; McCauley, John A; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J; DiMuzio, Jillian M; Ferrara, Marco; Filippo, Marcello Di; Gates, Adam T; Graham, Donald J; Harper, Steven; Hazuda, Daria J; Huang, Qian; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T; Soriano, Aileen; Stahlhut, Mark W; Vacca, Joseph P; Olsen, David B; Liverton, Nigel J; Carroll, Steven S

Discovery of 3-substituted aminocyclopentanes as potent and orally bioavailable NR2B subtype-selective NMDA antagonists

发现3-取代氨基环戊烷类化合物是高效且口服生物利用度高的NR2B亚型选择性NMDA拮抗剂

Layton, Mark E; Kelly, Michael J 3rd; Rodzinak, Kevin J; Sanderson, Philip E; Young, Steven D; Bednar, Rodney A; Dilella, Anthony G; McDonald, Terrence P; Wang, Hao; Mosser, Scott D; Fay, John F; Cunningham, Michael E; Reiss, Duane R; Fandozzi, Christine; Trainor, Nicole; Liang, Annie; Lis, Edward V; Seabrook, Guy R; Urban, Mark O; Yergey, James; Koblan, Kenneth S