日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

MeCP2 inhibits ischemic neuronal injury by enhancing methylation of the FOXO3a promoter to repress the SPRY2-ZEB1 axis

MeCP2 通过增强 FOXO3a 启动子甲基化来抑制 SPRY2-ZEB1 轴,从而抑制缺血性神经元损伤

Lei Meng, Bin Feng, Liming Luan, Zhihao Fang, Guangyu Zhao

Investigation of the structural requirements for N-methyl-D-aspartate receptor positive and negative allosteric modulators based on 2-naphthoic acid

基于2-萘甲酸的N-甲基-D-天冬氨酸受体正负变构调节剂的结构要求研究

Irvine, Mark W; Fang, Guangyu; Sapkota, Kiran; Burnell, Erica S; Volianskis, Arturas; Costa, Blaise M; Culley, Georgia; Collingridge, Graham L; Monaghan, Daniel T; Jane, David E

The NMDA receptor intracellular C-terminal domains reciprocally interact with allosteric modulators

NMDA受体胞内C端结构域与变构调节剂相互作用

Sapkota, Kiran; Dore, Kim; Tang, Kang; Irvine, Mark; Fang, Guangyu; Burnell, Erica S; Malinow, Roberto; Jane, David E; Monaghan, Daniel T

Dynamic generation of multi-qubit entanglement in the ultrastrong-coupling regime

在超强耦合机制下动态生成多量子比特纠缠

Liu, Xin; Liao, Qinghong; Fang, Guangyu; Liu, Shutian

The Startle Disease Mutation E103K Impairs Activation of Human Homomeric α1 Glycine Receptors by Disrupting an Intersubunit Salt Bridge across the Agonist Binding Site

惊吓病突变 E103K 通过破坏激动剂结合位点上的亚基间盐桥,损害人同源 α1 甘氨酸受体的激活。

Safar, Fatemah; Hurdiss, Elliot; Erotocritou, Marios; Greiner, Timo; Lape, Remigijus; Irvine, Mark W; Fang, Guangyu; Jane, David; Yu, Rilei; Dämgen, Marc A; Biggin, Philip C; Sivilotti, Lucia G

The NMDA receptor as a target for cognitive enhancement.

NMDA受体作为认知增强的靶点

Collingridge Graham L, Volianskis Arturas, Bannister Neil, France Grace, Hanna Lydia, Mercier Marion, Tidball Patrick, Fang Guangyu, Irvine Mark W, Costa Blaise M, Monaghan Daniel T, Bortolotto Zuner A, Molnár Elek, Lodge David, Jane David E

Piperazine-2,3-dicarboxylic acid derivatives as dual antagonists of NMDA and GluK1-containing kainate receptors

哌嗪-2,3-二羧酸衍生物作为NMDA和含GluK1的红藻氨酸受体的双重拮抗剂

Irvine, Mark W; Costa, Blaise M; Dlaboga, Daniel; Culley, Georgia R; Hulse, Richard; Scholefield, Caroline L; Atlason, Palmi; Fang, Guangyu; Eaves, Richard; Morley, Richard; Mayo-Martin, Maria B; Amici, Mascia; Bortolotto, Zuner A; Donaldson, Lucy; Collingridge, Graham L; Molnár, Elek; Monaghan, Daniel T; Jane, David E

Structure-activity relationships for allosteric NMDA receptor inhibitors based on 2-naphthoic acid

基于2-萘甲酸的变构NMDA受体抑制剂的构效关系

Costa, Blaise Mathias; Irvine, Mark W; Fang, Guangyu; Eaves, Richard J; Mayo-Martin, Maria Belen; Laube, Bodo; Jane, David E; Monaghan, Daniel T

Coumarin-3-carboxylic acid derivatives as potentiators and inhibitors of recombinant and native N-methyl-D-aspartate receptors

香豆素-3-羧酸衍生物作为重组和天然N-甲基-D-天冬氨酸受体的增强剂和抑制剂

Irvine, Mark W; Costa, Blaise M; Volianskis, Arturas; Fang, Guangyu; Ceolin, Laura; Collingridge, Graham L; Monaghan, Daniel T; Jane, David E

Pharmacological modulation of NMDA receptor activity and the advent of negative and positive allosteric modulators

NMDA受体活性的药理学调节以及负变构调节剂和正变构调节剂的出现

Monaghan, Daniel T; Irvine, Mark W; Costa, Blaise Mathias; Fang, Guangyu; Jane, David E