Profiling of drug resistance in Src kinase at scale uncovers a regulatory network coupling autoinhibition and catalytic domain dynamics.
大规模分析 Src 激酶的耐药性,揭示了一个将自身抑制和催化结构域动力学耦合起来的调控网络
期刊:Cell Chemical Biology
影响因子:7.2
doi:10.1016/j.chembiol.2023.08.005
Chakraborty Sujata, Ahler Ethan, Simon Jessica J, Fang Linglan, Potter Zachary E, Sitko Katherine A, Stephany Jason J, Guttman Miklos, Fowler Douglas M, Maly Dustin J