Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation
发现用于肿瘤治疗的高效选择性MTH1抑制剂:实现靶点(不)验证的快速开展
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.9b00420
Farand, Julie; Kropf, Jeffrey E; Blomgren, Peter; Xu, Jianjun; Schmitt, Aaron C; Newby, Zachary E; Wang, Ting; Murakami, Eisuke; Barauskas, Ona; Sudhamsu, Jawahar; Feng, Joy Y; Niedziela-Majka, Anita; Schultz, Brian E; Schwartz, Karen; Viatchenko-Karpinski, Serge; Kornyeyev, Dmytro; Kashishian, Adam; Fan, Peidong; Chen, Xiaowu; Lansdon, Eric B; Ports, Michael O; Currie, Kevin S; Watkins, William J; Notte, Gregory T