日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A trackable trinuclear platinum complex for breast cancer treatment.

一种用于乳腺癌治疗的可追踪三核铂配合物

O'Carroll Sinéad, Slator Creina, de Paiva Raphael E F, Newsome Conor, Searle Bethany, Kk Sriram, Whittle Sylvia, Catley Thomas E, Scoditti Stefano, Mnich Katarzyna, Peterson Erica J, Hu Bin, Koblinski Jennifer E, Samali Afshin, McKee Vickie, Pyne Alice L B, Westerlund Fredrik, Farrell Nicholas P, Kellett Andrew

Glycan Profiling Identifies Chondroitin-4-sulfate as a Biomarker for Platinum Response and Therapeutic Target in Ovarian Cancer

糖谱分析鉴定出硫酸软骨素-4是卵巢癌铂类药物疗效的生物标志物和治疗靶点

Peterson, Erica J; Hampton, James D; Weiss, Ryan J; Clausen, Thomas M; Beaudin, Ava R S; Deshmukh, Sharanya P; Dosmorov, Mikhail G; McGee Turner, Joseph B; Basu, Amrita; Vidal-Calvo, Elena Ethel; Daugard, Mads; Salanti, Ali; Koblinski, Jennifer E; Litovchick, Larisa; Farrell, Nicholas P

Probing Disaccharide Binding to Triplatin as Models for Tumor Cell Heparan Sulfate (GAG) Interactions

以二糖与三铂的结合为模型研究肿瘤细胞硫酸乙酰肝素(GAG)相互作用

Gorle, Anil K; Malde, Alpeshkumar K; Chang, Chih-Wei; Rajaratnam, Premraj; von Itzstein, Mark; Berners-Price, Susan J; Farrell, Nicholas P

A Click Chemistry Approach to Targeted DNA Crosslinking with cis-Platinum(II)-Modified Triplex-Forming Oligonucleotides

利用顺铂(II)修饰的三链形成寡核苷酸进行靶向DNA交联的点击化学方法

Hennessy, Joseph; McGorman, Bríonna; Molphy, Zara; Farrell, Nicholas P; Singleton, Daniel; Brown, Tom; Kellett, Andrew

Controlling Nuclease Degradation of Wireframe DNA Origami with Minor Groove Binders

利用小沟结合剂控制线框DNA折纸的核酸酶降解

Wamhoff, Eike-Christian; Romanov, Anna; Huang, Hellen; Read, Benjamin J; Ginsburg, Eric; Knappe, Grant A; Kim, Hyun Min; Farrell, Nicholas P; Irvine, Darrell J; Bathe, Mark

Exploitation of Sulfated Glycosaminoglycan Status for Precision Medicine of Triplatin in Triple-Negative Breast Cancer

利用硫酸糖胺聚糖状态进行三阴性乳腺癌三铂精准治疗

Hampton, James D; Peterson, Erica J; Katner, Samantha J; Turner, Tia H; Alzubi, Mohammad A; Harrell, J Chuck; Dozmorov, Mikhail G; Turner, Joseph B McGee; Gigliotti, Pam J; Kraskauskiene, Vita; Shende, Mayuri; Idowu, Michael O; Puchalapalli, Madhavi; Hu, Bin; Litovchick, Larisa; Katsuta, Eriko; Takabe, Kazuaki; Farrell, Nicholas P; Koblinski, Jennifer E

Molecular methods for assessment of non-covalent metallodrug-DNA interactions

评估非共价金属药物-DNA相互作用的分子方法

Kellett, Andrew; Molphy, Zara; Slator, Creina; McKee, Vickie; Farrell, Nicholas P

Substitution-inert trinuclear platinum complexes efficiently condense/aggregate nucleic acids and inhibit enzymatic activity

取代惰性的三核铂配合物能有效凝聚/聚集核酸并抑制酶活性。

Malina, Jaroslav; Farrell, Nicholas P; Brabec, Viktor

Dinuclear platinum complexes containing planar aromatic ligands to enhance stacking interactions with proteins

含有平面芳香配体的双核铂配合物可增强与蛋白质的堆积相互作用

Ma, Erin S F; Daniel, A Gerard; Farrell, Nicholas P

Retained platinum uptake and indifference to p53 status make novel transplatinum agents active in platinum-resistant cells compared to cisplatin and oxaliplatin

与顺铂和奥沙利铂相比,新型反式铂类药物由于保留了铂的摄取能力且不受p53状态的影响,因此对铂耐药细胞具有活性。

Murphy, Robert F; Komlodi-Pasztor, Edina; Robey, Robert; Balis, Frank M; Farrell, Nicholas P; Fojo, Tito