日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mechanistic insights into the therapeutic properties of delta opioid receptor

对δ阿片受体治疗特性的机制性见解

Bernhard, Sarah M; Roy Chowdhury, Susovan; Murata, Tsuyoshi; Reinl, Erin L; Ramos-Gonzalez, Nokomis; Denn, Elizabeth; Appourchaux, Kevin; Inoue, Asuka; England, Sarah K; Fay, Jonathan F; Majumdar, Susruta; Chanda, Baron; Che, Tao

The structural diversity of psychedelic drug actions revealed

迷幻药作用的结构多样性揭示

Gumpper, Ryan H; Jain, Manish K; Kim, Kuglae; Sun, Renhong; Sun, Ning; Xu, Zhongli; DiBerto, Jeffrey F; Krumm, Brian E; Kapolka, Nicholas J; Kaniskan, H Ümit; Nichols, David E; Jin, Jian; Fay, Jonathan F; Roth, Bryan L

Structure-guided design of partial agonists at an opioid receptor.

基于结构的阿片受体部分激动剂设计

Varga Balazs R, Bernhard Sarah M, El Daibani Amal, Zaidi Saheem A, Lam Jordy H, Aguilar Jhoan, Appourchaux Kevin, Nazarova Antonina L, Kouvelis Alexa, Shinouchi Ryosuke, Hammond Haylee R, Eans Shainnel O, Weinreb Violetta, Margolis Elyssa B, Fay Jonathan F, Huang Xi-Ping, Pradhan Amynah, Katritch Vsevolod, McLaughlin Jay P, Majumdar Susruta, Che Tao

Structure of human green cone opsin yields insights into mechanisms underlying the rapid decay of its active, signaling state

人类绿色视锥细胞视蛋白的结构揭示了其活性信号状态快速衰减的机制。

Yao, Weekie; Fay, Jonathan F; Farrens, David L

UDP-glucose and MRS2905 agonist-bound states of the purinergic P2Y(14) receptor

嘌呤能P2Y(14)受体的UDP-葡萄糖和MRS2905激动剂结合状态

Fay, Jonathan F; Kousouros, Joseph; Gao, Zhan-Guo; Pavan, Matteo; Oliva, Paola; Pramanik, Asmita; Meyer, Clayton; Kurma, Siva Hariprasad; Xu, Wen; Krumm, Brian; Jacobson, Kenneth A

Structure-guided design of a peripherally restricted chemogenetic system.

结构导向的外周限制性化学遗传系统设计

Kang Hye Jin, Krumm Brian E, Tassou Adrien, Geron Matan, DiBerto Jeffrey F, Kapolka Nicholas J, Gumpper Ryan H, Sakamoto Kensuke, Dewran Kocak D, Olsen Reid H J, Huang Xi-Ping, Zhang Shicheng, Huang Karen L, Zaidi Saheem A, Nguyen MyV T, Jo Min Jeong, Katritch Vsevolod, Fay Jonathan F, Scherrer Grégory, Roth Bryan L

MRGPRX4 mediates phospho-drug-associated pruritus in a humanized mouse model

MRGPRX4介导人源化小鼠模型中磷酸化药物相关的瘙痒

Chien, Daphne Chun-Che; Limjunyawong, Nathachit; Cao, Can; Meixiong, James; Peng, Qi; Ho, Cheng-Ying; Fay, Jonathan F; Roth, Bryan L; Dong, Xinzhong

High-affinity agonists reveal recognition motifs for the MRGPRD GPCR.

高亲和力激动剂揭示了 MRGPRD GPCR 的识别基序

Wang Chunyu, Liu Yongfeng, Lanier Marion, Yeager Adam, Singh Isha, Gumpper Ryan H, Krumm Brian E, DeLeon Chelsea, Zhang Shicheng, Boehm Marcus, Pittner Richard, Baron Alain, Dvorak Lisa, Bacon Corinne, Shoichet Brian K, Martinborough Esther, Fay Jonathan F, Cao Can, Roth Bryan L

High-speed high-resolution data collection on a 200 keV cryo-TEM

在200 keV冷冻透射电镜上进行高速高分辨率数据采集。

Peck, Jared V; Fay, Jonathan F; Strauss, Joshua D

Single Proteoliposome High-Content Analysis Reveals Differences in the Homo-Oligomerization of GPCRs

单蛋白脂质体高内涵分析揭示GPCR同源寡聚化的差异

Walsh, Samuel M; Mathiasen, Signe; Christensen, Sune M; Fay, Jonathan F; King, Christopher; Provasi, Davide; Borrero, Ernesto; Rasmussen, Søren G F; Fung, Juan Jose; Filizola, Marta; Hristova, Kalina; Kobilka, Brian; Farrens, David L; Stamou, Dimitrios