日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tumor-Targeted Delivery of an EGFR Inhibitor Prodrug via Site-Specific Albumin Conjugation

通过位点特异性白蛋白偶联将 EGFR 抑制剂前药靶向递送至肿瘤部位

Federa, Anja; Pitek, Rastislav; Dömötör, Orsolya; Enyedy, Éva A; Terenzi, Alessio; Caban, Monika; Stefanelli, Alessia; D'Anna, Luisa; White, Faye; Heffeter, Petra; Kowol, Christian R

Site-Selectively Functionalized Albumin with DFO*Maleimide for (89)Zr-Radiolabeling Yields a Metabolically Stable PET Probe that Enables Late Time-Point Tumor Imaging in Mice.

用 DFO*马来酰亚胺对白蛋白进行位点选择性功能化,用于 (89)Zr 放射性标记,可产生代谢稳定的 PET 探针,从而实现小鼠的晚期肿瘤成像

Kronberger Julia, Balber Theresa, Schueffl Hemma, Wahrmann Raphaela, Federa Anja, Gradl Mathias, Brandt Marie R, Wanek Thomas, Mitterhauser Markus, Kowol Christian R, Mindt Thomas L, Heffeter Petra

A new fluorescent oxaliplatin(iv) complex with EGFR-inhibiting properties for the treatment of drug-resistant cancer cells

一种新型荧光奥沙利铂(IV)复合物,具有EGFR抑制特性,可用于治疗耐药癌细胞。

Caban, Monika; Fronik, Philipp; Terenzi, Alessio; Federa, Anja; Bormio Nunes, Julia H; Pitek, Rastislav; Kirchhofer, Dominik; Schueffl, Hemma H; Berger, Walter; Keppler, Bernhard K; Kowol, Christian R; Heffeter, Petra

Novel Maleimide Linkers Based on a Piperazine Motif for Strongly Increased Aqueous Solubility

基于哌嗪基团的新型马来酰亚胺连接剂可显著提高水溶性

Dijkstra, Martijn; Schueffl, Hemma; Federa, Anja; Kast, Caroline; Unterlercher, Alexander; Keppler, Bernhard K; Heffeter, Petra; Kowol, Christian R

Comparative Evaluation of Thiol- and Amine-Conjugating Moieties for Endogenous Albumin Binding after Intravenous Administration.

静脉注射后硫醇和胺结合部分与内源性白蛋白结合的比较评价

Federa Anja, Schueffl Hemma, Minichmayr Iris K, Kastner Alexander, Kronberger Julia, Mindt Thomas L, Heffeter Petra, Kowol Christian R