日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Proteogenomic investigation of plant constituents in herbal beverages

草本饮料中植物成分的蛋白质组学研究

Chudinov, Ivan K; Krinitsina, Anastasia A; Petukhova, Diana A; Lukina-Gronskaya, Aleksandra V; Korneenko, Elena V; Gremyacheva, Veronika D; Kovalenko, Alexey V; Fedorov, Oleg V; Kozhemyakin, Grigory L; Mironov, Kirill S; Antipin, Maxim I; Butenko, Ivan O; Logacheva, Maria D; Speranskaya, Anna S

Binding-Site Purification of Actives (B-SPA) Enables Efficient Large-Scale Progression of Fragment Hits by Combining Multi-Step Array Synthesis With HT Crystallography

结合位点活性化合物纯化(B-SPA)结合多步阵列合成和高通量晶体学,可实现片段先导化合物的高效大规模筛选。

Grosjean, Harold; Aimon, Anthony; Hassell-Hart, Storm; Thompson, Warren; Koekemoer, Lizbé; Bennett, James; Bradley, Anthony; Anderson, Cameron; Wild, Conor; Bradshaw, William J; FitzGerald, Edward A; Krojer, Tobias; Fedorov, Oleg; Biggin, Philip C; Spencer, John; von Delft, Frank

Structure-Guided Design of ISOX-DUAL-Based Degraders Targeting BRD4 and CBP/EP300: A Case of Degrader Collapse.

基于 ISOX-DUAL 的结构导向降解剂设计:针对 BRD4 和 CBP/EP300 的降解剂崩溃案例

Edmonds Anthony K, Balourdas Dimitrios-Ilias, Marsh Graham P, Felix Robert, Brasher Bradley, Cooper Jeff, Graber-Feesl Cari, Kollareddy Madhu, Malik Karim, Stewart Helen, Chevassut Timothy J T, Lineham Ella, Morley Simon, Fedorov Oleg, Bennett James, Rajasekaran Mohan B, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Joerger Andreas C, Maple Hannah J, Spencer John

SARS-CoV-2 FP1 Destabilizes Lipid Membranes and Facilitates Pore Formation

SARS-CoV-2 FP1 破坏脂质膜并促进孔道形成

Sumarokova, Maria; Pavlov, Rais; Lavushchenko, Tatiana; Vasilenko, Egor; Kozhemyakin, Grigory; Fedorov, Oleg; Molotkovsky, Rodion; Bashkirov, Pavel

Antibiotic resistance and viral co-infection in children diagnosed with pneumonia caused by Mycoplasma pneumoniae admitted to Russian hospitals during October 2023-February 2024

2023年10月至2024年2月期间,俄罗斯医院收治的由肺炎支原体引起的肺炎患儿的抗生素耐药性和病毒合并感染情况

Korneenko, Elena; Rog, Irina; Chudinov, Ivan; Lukina-Gronskaya, Aleksandra; Kozyreva, Anfisa; Belyaletdinova, Ilmira; Kuzmina, Julia; Fedorov, Oleg; Evsyutina, Daria; Shunaev, Alexey; Matyushkina, Daria; Govorun, Vadim; Speranskaya, Anna

Interaction of two strongly divergent archaellins stabilizes the structure of the Halorubrum archaellum

两种差异极大的古菌素相互作用稳定了盐红古菌的结构。

Pyatibratov, Mikhail G; Syutkin, Alexey S; Quax, Tessa E F; Melnik, Tatjana N; Papke, R Thane; Gogarten, Johann Peter; Kireev, Igor I; Surin, Alexey K; Beznosov, Sergei N; Galeva, Anna V; Fedorov, Oleg V

An Activity-Based Probe Targeting Non-Catalytic, Highly Conserved Amino Acid Residues within Bromodomains

一种靶向溴结构域内非催化性、高度保守氨基酸残基的活性探针

D'Ascenzio, Melissa; Pugh, Kathryn M; Konietzny, Rebecca; Berridge, Georgina; Tallant, Cynthia; Hashem, Shaima; Monteiro, Octovia; Thomas, Jason R; Schirle, Markus; Knapp, Stefan; Marsden, Brian; Fedorov, Oleg; Bountra, Chas; Kessler, Benedikt M; Brennan, Paul E

Design, Synthesis and Characterization of Covalent KDM5 Inhibitors

共价KDM5抑制剂的设计、合成和表征

Vazquez-Rodriguez, Saleta; Wright, Miranda; Rogers, Catherine M; Cribbs, Adam P; Velupillai, Srikannathasan; Philpott, Martin; Lee, Henry; Dunford, James E; Huber, Kilian V M; Robers, Matthew B; Vasta, James D; Thezenas, Marie-Laetitia; Bonham, Sarah; Kessler, Benedikt; Bennett, James; Fedorov, Oleg; Raynaud, Florence; Donovan, Adam; Blagg, Julian; Bavetsias, Vassilios; Oppermann, Udo; Bountra, Chas; Kawamura, Akane; Brennan, Paul E

Salt-dependent regulation of archaellins in Haloarcula marismortui

盐依赖性调控在死海盐弧菌(Haloarcula marismortui)中古生菌素的表达

Syutkin, Alexey S; van Wolferen, Marleen; Surin, Alexey K; Albers, Sonja-Verena; Pyatibratov, Mikhail G; Fedorov, Oleg V; Quax, Tessa E F

Discovery of an MLLT1/3 YEATS Domain Chemical Probe

MLLT1/3 YEATS结构域化学探针的发现

Moustakim, Moses; Christott, Thomas; Monteiro, Octovia P; Bennett, James; Giroud, Charline; Ward, Jennifer; Rogers, Catherine M; Smith, Paul; Panagakou, Ioanna; Díaz-Sáez, Laura; Felce, Suet Ling; Gamble, Vicki; Gileadi, Carina; Halidi, Nadia; Heidenreich, David; Chaikuad, Apirat; Knapp, Stefan; Huber, Kilian V M; Farnie, Gillian; Heer, Jag; Manevski, Nenad; Poda, Gennady; Al-Awar, Rima; Dixon, Darren J; Brennan, Paul E; Fedorov, Oleg