日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Covalent Inhibitors of KEAP1 with Exquisite Selectivity.

具有极高选择性的KEAP1共价抑制剂

Fejes Imre, Markacz Piroska, Tatai Janos, Rudas Monika, Dunkel Petra, Gyuris Mario, Nyerges Miklos, Provost Nicolas, Duvivier Valérie, Delerive Philippe, Martiny Virginie, Bristiel Alexandra, Vidal Brice, Richardson William, Rothweiler Elisabeth M, Tranberg-Jensen Jeppe, Manning Charlotte E, Sweeney Melissa N, Chalk Rod, Huber Kilian V M, Bullock Alex N, Herner Andras, Seedorf Klaus, Vinson Cedric, Weber Csaba, Kotschy Andras

Targeting NOX2 via p47/phox-p22/phox Inhibition with Novel Triproline Mimetics

利用新型三脯氨酸模拟物通过抑制p47/phox-p22/phox靶向NOX2

Garsi, Jean-Baptiste; Komjáti, Balázs; Cullia, Gregorio; Fejes, Imre; Sipos, Melinda; Sipos, Zoltán; Fördős, Eszter; Markacz, Piroska; Balázs, Barbara; Lancelot, Nathalie; Berger, Sylvie; Raimbaud, Eric; Brown, David; Vuillard, Laurent-Michel; Haberkorn, Laure; Cukier, Cyprian; Szlávik, Zoltán; Hanessian, Stephen