日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Guided Design of ISOX-DUAL-Based Degraders Targeting BRD4 and CBP/EP300: A Case of Degrader Collapse.

基于 ISOX-DUAL 的结构导向降解剂设计:针对 BRD4 和 CBP/EP300 的降解剂崩溃案例

Edmonds Anthony K, Balourdas Dimitrios-Ilias, Marsh Graham P, Felix Robert, Brasher Bradley, Cooper Jeff, Graber-Feesl Cari, Kollareddy Madhu, Malik Karim, Stewart Helen, Chevassut Timothy J T, Lineham Ella, Morley Simon, Fedorov Oleg, Bennett James, Rajasekaran Mohan B, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Joerger Andreas C, Maple Hannah J, Spencer John

Except for Robust Outliers, Rapamycin Increases Lesion Burden in a Murine Model of Cerebral Cavernous Malformations

除稳健的异常值外,雷帕霉素会增加小鼠脑海绵状血管畸形模型中的病变负担

Roberto J Alcazar-Felix, Robert Shenkar, Christian R Benavides, Akash Bindal, Abhinav Srinath, Ying Li, Serena Kinkade, Tatiana Terranova, Evon DeBose-Scarlett, Rhonda Lightle, Dorothy DeBiasse, Hanadi Almazroue, Diana Vera Cruz, Sharbel Romanos, Aditya Jhaveri, Janne Koskimäki, Stephanie Hage, Caro

Vitamin B2 enables regulation of fasting glucose availability

维生素 B2 能够调节空腹血糖的利用率

Peter M Masschelin, Pradip Saha, Scott A Ochsner, Aaron R Cox, Kang Ho Kim, Jessica B Felix, Robert Sharp, Xin Li, Lin Tan, Jun Hyoung Park, Liping Wang, Vasanta Putluri, Philip L Lorenzi, Alli M Nuotio-Antar, Zheng Sun, Benny Abraham Kaipparettu, Nagireddy Putluri, David D Moore, Scott A Summers, N

The rheumatoid arthritis drug auranofin lowers leptin levels and exerts antidiabetic effects in obese mice

类风湿性关节炎药物金诺芬可降低肥胖小鼠的瘦素水平并发挥抗糖尿病作用。

Aaron R Cox ,Peter M Masschelin ,Pradip K Saha ,Jessica B Felix ,Robert Sharp ,Zeqin Lian ,Yan Xia ,Natasha Chernis ,David A Bader ,Kang Ho Kim ,Xin Li ,Jun Yoshino ,Xin Li ,Gang Li ,Zheng Sun ,Huaizhu Wu ,Cristian Coarfa ,David D Moore ,Samuel Klein ,Kai Sun ,Sean M Hartig

Developing degraders: principles and perspectives on design and chemical space

降解剂的开发:设计和化学空间的原则和视角

Maple, Hannah J; Clayden, Nat; Baron, Anne; Stacey, Callum; Felix, Robert

Hydrogen/deuterium exchange mass spectrometry and computational modeling reveal a discontinuous epitope of an antibody/TL1A Interaction

氢/氘交换质谱和计算建模揭示了抗体/TL1A 相互作用的不连续表位

Richard Y-C Huang, Stanley R Krystek Jr, Nathan Felix, Robert F Graziano, Mohan Srinivasan, Achal Pashine, Guodong Chen

N 1-Arylation of 1,4-Benzodiazepine-2-ones with Diaryliodonium Salts

用二芳基碘鎓盐对 1,4-苯并二氮杂卓-2-酮进行 N 1-芳基化

Shim, Eunjae; Zakarian, Armen; Khan, Raysa; Felix, Robert; Kemmitt, Paul D; Coles, Simon J; Tizzard, Graham J; Spencer, John

Combining Sanford Arylations on Benzodiazepines with the Nuisance Effect

将桑福德芳基化修饰苯二氮卓类药物与干扰效应相结合

Khan, Raysa; Boonseng, Sarote; Kemmitt, Paul D; Felix, Robert; Coles, Simon J; Tizzard, Graham J; Williams, Gareth; Simmonds, Olivia; Harvey, Jessica-Lily; Atack, John; Cox, Hazel; Spencer, John

Using the electronic medical record to refer women taking category D or X medications for teratogen and contraceptive counseling

利用电子病历将服用D类或X类药物的女性转诊至致畸剂和避孕咨询机构。

Mody, Sheila K; Wu, Jennifer; Ornelas, Marla; Kernahan, Colleen; Salas, Elizabeth; Kao, Kelly; Felix, Robert; Chambers, Christina

Using the electronic medical record to assess contraception usage among women taking category D or X medications

利用电子病历评估服用D类或X类药物的女性的避孕措施使用情况

Mody, Sheila K; Farala, John Paul; Wu, Jennifer; Felix, Robert; Chambers, Christina