日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Metal-polyphenol network-based multifunctional materials for tumor therapy: Intrinsic properties, advances, and applications

基于金属-多酚网络的多功能材料在肿瘤治疗中的应用:固有特性、研究进展及应用

Ma, Chen; Xu, Qian; Ding, Lingwen; Liu, Xinya; Cheng, Junkai; Wang, Yiman; Liu, Lu; Xian, Jiaqi; Gu, Jian; Tran, Phuong-Thao; Wang, Qin; Wang, Shuai; Chen, Fen-Er

Discovery of novel coumarin-containing triazolo[1,5-a]pyrimidine derivatives as potent ABCB1 inhibitor for modulation of multidrug resistance.

发现新型含香豆素的三唑并[1,5-a]嘧啶衍生物作为强效ABCB1抑制剂,用于调节多药耐药性。

Hmone Nan Ye, Tian Xuefei, Zhou Dandan, Min Zhiyi, Zhao Yingxue, Wang Shuai, Chen Fen-Er, Wang Ziyu, Zhang Xuyao

Bioisosterism-driven design of orally active, safe, and broad-spectrum biphenyl-DAPY derivatives as highly potent HIV-1 non-nucleoside reverse transcriptase inhibitors

基于生物等排效应设计的口服活性、安全、广谱联苯-DAPY衍生物作为高效的HIV-1非核苷类逆转录酶抑制剂

Chen, Xiao-Mei; Hao, Qing-Qing; Pannecouque, Christophe; De Clercq, Erik; Wang, Shuai; Chen, Fen-Er

Enhancing Reaction Compatibility in Telescoped Multistep Flow Synthesis via Hybridizing Micro Packed-Bed/Micro Tubing Reactors: Application to Cyproflanilide and Broflanilide

通过混合微型填充床/微型管式反应器增强串联多步流动合成的反应兼容性:以环丙苯胺和溴苯胺为例

Zhang, Xingyu; Huang, Gangqin; Ou, Yihui; Luo, Zeyi; Huang, Zheyao; Liu, Chenguang; Chen, Fen-Er

Picomolar inhibitor of reverse transcriptase featuring significantly improved metabolic stability

皮摩尔级逆转录酶抑制剂,具有显著提高的代谢稳定性

Sang, Ya-Li; Pannecouque, Christophe; De Clercq, Erik; Wang, Shuai; Chen, Fen-Er

Structure-based design of novel heterocycle-substituted ATDP analogs as non-nucleoside reverse transcriptase inhibitors with improved selectivity and solubility

基于结构的新型杂环取代ATDP类似物设计,作为具有更高选择性和溶解度的非核苷类逆转录酶抑制剂

Zhao, Li-Min; Pannecouque, Christophe; Clercq, Erik De; Wang, Shuai; Chen, Fen-Er

Highly enantioselective synthesis of both tetrahydroquinoxalines and dihydroquinoxalinones via Rh-thiourea catalyzed asymmetric hydrogenation

通过铑-硫脲催化的不对称氢化反应,高对映选择性地合成四氢喹喔啉和二氢喹喔啉酮。

Xu, Ana; Li, Chaoyi; Huang, Junrong; Pang, Heng; Zhao, Chengyao; Song, Lijuan; You, Hengzhi; Zhang, Xumu; Chen, Fen-Er

Recent development on COX-2 inhibitors as promising anti-inflammatory agents: The past 10 years

COX-2 抑制剂作为有前途的抗炎药物的最新进展:过去 10 年

Zhiran Ju, Menglan Li, Junde Xu, Daniel C Howell, Zhiyun Li, Fen-Er Chen

Construction of Non-Biaryl Atropisomeric Amide Scaffolds Bearing a C-N Axis via Enantioselective Catalysis

通过对映选择性催化构建带有CN轴的非联芳基阻转异构酰胺骨架

Xiao, Xiao; Chen, Biao; Yao, Yi-Ping; Zhou, Hai-Jie; Wang, Xu; Wang, Neng-Zhong; Chen, Fen-Er

Synthesis and Evaluation of NF-κB Inhibitory Activity of Mollugin Derivatives

Mollugin衍生物的合成及NF-κB抑制活性评价

Lin-Hao Zhang, Ming-Yue Li, Da-Yuan Wang, Xue-Jun Jin, Fen-Er Chen, Hu-Ri Piao