日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

1'- and 4'-Cyano Modified Adenosine Analogs Against Prototypic Flavivirus RNA-Dependent RNA Polymerases

1'-和4'-氰基修饰的腺苷类似物对抗原型黄病毒RNA依赖性RNA聚合酶

Walker, Simon M; Gordon, Calvin J; Tchesnokov, Egor P; Sun, Long; Zou, Jing; Xie, Xuping; Riola, Nicholas C; Cutillas, Vincent; Du Pont, Venice; Zhao, Xiaofeng; Wang, Ting; Pitts, Jared; Siegel, Dustin S; Perry, Jason K; Feng, Joy Y; Bilello, John P; Götte, Matthias

Meeting report: 38th international conference on antiviral research in Las Vegas, United States of America, March 17-21, 2025

会议报告:第38届国际抗病毒研究大会,美国拉斯维加斯,2025年3月17日至21日

Jordan, Robert; Archin, Nancie M; Cagno, Valeria; Feng, Joy Y; Guo, Haitao; Herrero, Lara J; Janeba, Zlatko; Meanwell, Nicholas A; Moffat, Jennifer; Neyts, Johan; Rocha-Pereira, Joana; Seley-Radtke, Kathie L; Sheahan, Timothy P; Spengler, Jessica R; Welch, Stephen R; Xie, Xuping; Zakaryan, Hovakim; Schang, Luis M; Durantel, David

Template switching by coronavirus polymerase requires helicase activity and is stimulated by remdesivir and molnupiravir

冠状病毒聚合酶的模板转换需要解旋酶活性,并可被瑞德西韦和莫努皮韦刺激。

Rakib, Asif; Das, Arnab; Bera, Subhas C; America, Pim P B; Klein, Misha; Anderson, Thomas K; Marecki, John C; Wang, Bing; Bogers, Eline; Feng, Joy Y; Bilello, John P; Papini, Flávia S; Smitskamp, Quinte; Arnold, Jamie J; Artsimovitch, Irina; Kirchdoerfer, Robert N; Cameron, Craig E; Raney, Kevin D; Dulin, David

Meeting report of the 37th International Conference on Antiviral Research in Gold Coast, Australia, May 20-24, 2024, organized by the International Society for Antiviral Research

第37届国际抗病毒研究大会会议报告,2024年5月20日至24日,澳大利亚黄金海岸,由国际抗病毒研究学会主办

Welch, Stephen R; Bilello, John P; Carter, Kara; Delang, Leen; Dirr, Larissa; Durantel, David; Feng, Joy Y; Gowen, Brian B; Herrero, Lara J; Janeba, Zlatko; Kleymann, Gerald; Lee, Alpha A; Meier, Chris; Moffat, Jennifer; Schang, Luis M; Schiffer, Joshua T; Seley-Radtke, Katherine L; Sheahan, Timothy P; Spengler, Jessica R

Interfering with nucleotide excision by the coronavirus 3'-to-5' exoribonuclease

干扰冠状病毒 3' 至 5' 外切核糖核酸酶的核苷酸切除

Chinthapatla, Rukesh; Sotoudegan, Mohamad; Srivastava, Pankaj; Anderson, Thomas K; Moustafa, Ibrahim M; Passow, Kellan T; Kennelly, Samantha A; Moorthy, Ramkumar; Dulin, David; Feng, Joy Y; Harki, Daniel A; Kirchdoerfer, Robert N; Cameron, Craig E; Arnold, Jamie J

Efficacy of the oral nucleoside prodrug GS-5245 (Obeldesivir) against SARS-CoV-2 and coronaviruses with pandemic potential

口服核苷前药GS-5245(奥贝地西韦)对SARS-CoV-2和具有大流行潜力的冠状病毒的疗效

Martinez, David R; Moreira, Fernando R; Zweigart, Mark R; Gully, Kendra L; De la Cruz, Gabriela; Brown, Ariane J; Adams, Lily E; Catanzaro, Nicholas; Yount, Boyd; Baric, Thomas J; Mallory, Michael L; Conrad, Helen; May, Samantha R; Dong, Stephanie; Scobey, D Trevor; Montgomery, Stephanie A; Perry, Jason; Babusis, Darius; Barrett, Kimberly T; Nguyen, Anh-Hoa; Nguyen, Anh-Quan; Kalla, Rao; Bannister, Roy; Bilello, John P; Feng, Joy Y; Cihlar, Tomas; Baric, Ralph S; Mackman, Richard L; Schäfer, Alexandra; Sheahan, Timothy P

An atomistic model of the coronavirus replication-transcription complex as a hexamer assembled around nsp15

冠状病毒复制转录复合物的原子模型,该复合物是由nsp15组装而成的六聚体。

Perry, Jason K; Appleby, Todd C; Bilello, John P; Feng, Joy Y; Schmitz, Uli; Campbell, Elizabeth A

Correction: Template-dependent inhibition of coronavirus RNA-dependent RNA polymerase by remdesivir reveals a second mechanism of action

更正:瑞德西韦对冠状病毒RNA依赖性RNA聚合酶的模板依赖性抑制揭示了其第二种作用机制

Tchesnokov, Egor P; Gordon, Calvin J; Woolner, Emma; Kocincova, Dana; Perry, Jason K; Feng, Joy Y; Porter, Danielle P; Götte, Matthias

Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation

发现用于肿瘤治疗的高效选择性MTH1抑制剂:实现靶点(不)验证的快速开展

Farand, Julie; Kropf, Jeffrey E; Blomgren, Peter; Xu, Jianjun; Schmitt, Aaron C; Newby, Zachary E; Wang, Ting; Murakami, Eisuke; Barauskas, Ona; Sudhamsu, Jawahar; Feng, Joy Y; Niedziela-Majka, Anita; Schultz, Brian E; Schwartz, Karen; Viatchenko-Karpinski, Serge; Kornyeyev, Dmytro; Kashishian, Adam; Fan, Peidong; Chen, Xiaowu; Lansdon, Eric B; Ports, Michael O; Currie, Kevin S; Watkins, William J; Notte, Gregory T

Nucleotide Prodrug Containing a Nonproteinogenic Amino Acid To Improve Oral Delivery of a Hepatitis C Virus Treatment

含有非蛋白源性氨基酸的核苷酸前药可改善丙型肝炎病毒治疗药物的口服递送

Feng, Joy Y; Wang, Ting; Park, Yeojin; Babusis, Darius; Birkus, Gabriel; Xu, Yili; Voitenleitner, Christian; Fenaux, Martijn; Yang, Huiling; Eng, Stacey; Tirunagari, Neeraj; Kirschberg, Thorsten; Cho, Aesop; Ray, Adrian S