日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Humanization of Drug Metabolism in the Plasmodium berghei Mouse Model for Antimalarial Drug Discovery

利用伯氏疟原虫小鼠模型进行药物代谢人源化研究以开发抗疟药物

MacLeod, A Kenneth; Merino, Cristina; Viera-Morilla, Sara; Frame, Laura; Tavendale, Amy; Duncan, Christina; Ferguson, Liam; Pinto, Erika G; Simeons, Frederick R C; Gomez-Jimenez, Vanessa; García, Ana Belén; Riley, Jennifer; Shishikura, Yoko; Martínez-Martínez, María Santos; Wolf, C Roland; Read, Kevin D

Cryptosporidium lysyl-tRNA synthetase inhibitors define the interplay between solubility and permeability required to achieve efficacy

隐孢子虫赖氨酰tRNA合成酶抑制剂阐明了溶解度和渗透性之间的相互作用,而这种相互作用是实现疗效所必需的。

Caldwell, Nicola; Peet, Caroline; Miller, Peter; Colon, Beatrice L; Taylor, Malcolm G; Cocco, Mattia; Dawson, Alice; Lukac, Iva; Teixeira, Jose E; Robinson, Lee; Frame, Laura; Seizova, Simona; Damerow, Sebastian; Tamaki, Fabio; Post, John; Riley, Jennifer; Mutter, Nicole; Hanna, Jack C; Ferguson, Liam; Hu, Xiao; Tinti, Michele; Forte, Barbara; Norcross, Neil R; Campbell, Peter S; Svensen, Nina; Caldwell, Flora C; Jansen, Chimed; Postis, Vincent; Read, Kevin D; Huston, Christopher D; Gilbert, Ian H; Baragaña, Beatriz; Pawlowic, Mattie C

Rational Exploration of 2,4-Diaminopyrimidines as DHFR Inhibitors Active against Mycobacterium abscessus and Mycobacterium avium, Two Emerging Human Pathogens.

合理探索 2,4-二氨基嘧啶作为 DHFR 抑制剂对脓肿分枝杆菌和鸟分枝杆菌(两种新兴人类病原体)的活性

Andrade Meirelles Matheus, Almeida Vitor M, Sullivan Jaryd R, de Toledo Ian, Dos Reis Caio Vinicius, Cunha Micael Rodrigues, Zigweid Rachel, Shim Abraham, Sankaran Banumathi, Woodward Elijah L, Seibold Steve, Liu Lijun, Mian Mohammad Rasel, Battaile Kevin P, Riley Jennifer, Duncan Christina, Simeons Frederick R C, Ferguson Liam, Joji Halimatu, Read Kevin D, Lovell Scott, Staker Bart L, Behr Marcel A, Pilli Ronaldo A, Couñago Rafael M

Microplastic concentrations and risk assessment in water, sediment and invertebrates from Simon's Town, South Africa

南非西蒙镇水体、沉积物和无脊椎动物中微塑料浓度及风险评估

Ferguson, Liam; Awe, Adetunji; Sparks, Conrad

Identification and development of a series of disubstituted piperazines for the treatment of Chagas disease

鉴定和开发一系列二取代哌嗪类化合物用于治疗恰加斯病

McGonagle, Kate; Tarver, Gary J; Cantizani, Juan; Cotillo, Ignacio; Dodd, Peter G; Ferguson, Liam; Gilbert, Ian H; Marco, Maria; Miles, Tim; Naylor, Claire; Osuna-Cabello, Maria; Paterson, Christy; Read, Kevin D; Pinto, Erika G; Riley, Jennifer; Scullion, Paul; Shishikura, Yoko; Simeons, Frederick; Stojanovski, Laste; Svensen, Nina; Thomas, John; Wyatt, Paul G; Manzano, Pilar; De Rycker, Manu; Thomas, Michael G