日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemical Proteomics Reveals Off-Targets of the Anandamide Reuptake Inhibitor WOBE437

化学蛋白质组学揭示花生四烯乙醇胺再摄取抑制剂 WOBE437 的脱靶效应

Berend Gagestein, Anna F Stevens, Domenico Fazio, Bogdan I Florea, Tom van der Wel, Alexander T Bakker, Filomena Fezza, Hans den Dulk, Herman S Overkleeft, Mauro Maccarrone, Mario van der Stelt

In Silico and In Vitro Analysis of Major Cannabis-Derived Compounds as Fatty Acid Amide Hydrolase Inhibitors

对主要大麻衍生化合物作为脂肪酸酰胺水解酶抑制剂的计算机模拟和体外分析

Emanuele Criscuolo, Maria Laura De Sciscio, Filomena Fezza, Mauro Maccarrone

Bisphenol A Deranges the Endocannabinoid System of Primary Sertoli Cells with an Impact on Inhibin B Production

双酚 A 扰乱原代塞托利细胞的内源性大麻素系统,影响抑制素 B 的产生

Gianna Rossi, Beatrice Dufrusine, Anna Rita Lizzi, Carla Luzi, Alessandra Piccoli, Filomena Fezza, Roberto Iorio, Gabriele D'Andrea, Enrico Dainese, Sandra Cecconi, Mauro Maccarrone

Cannabinoid CB2 receptor ligand profiling reveals biased signalling and off-target activity

大麻素 CB2 受体配体分析揭示了偏向信号和脱靶活性

Marjolein Soethoudt, Uwe Grether, Jürgen Fingerle, Travis W Grim, Filomena Fezza, Luciano de Petrocellis, Christoph Ullmer, Benno Rothenhäusler, Camille Perret, Noortje van Gils, David Finlay, Christa MacDonald, Andrea Chicca, Marianela Dalghi Gens, Jordyn Stuart, Henk de Vries, Nicolina Mastrangelo

Lipid Discovery by Combinatorial Screening and Untargeted LC-MS/MS

通过组合筛选和非靶向 LC-MS/MS 发现脂质

Mesut Bilgin, Petra Born, Filomena Fezza, Michael Heimes, Nicolina Mastrangelo, Nicolai Wagner, Carsten Schultz, Mauro Maccarrone, Suzanne Eaton, André Nadler, Matthias Wilm, Andrej Shevchenko

Endocannabinoids, related compounds and their metabolic routes

内源性大麻素、相关化合物及其代谢途径

Filomena Fezza, Monica Bari, Rita Florio, Emanuela Talamonti, Monica Feole, Mauro Maccarrone

Activation of type-2 cannabinoid receptor inhibits neuroprotective and antiinflammatory actions of glucocorticoid receptor α: when one is better than two

型大麻素受体的激活会抑制糖皮质激素受体 α 的神经保护和抗炎作用:一种优于两种

Elisa Bisicchia, Valerio Chiurchiù, Maria Teresa Viscomi, Laura Latini, Filomena Fezza, Luca Battistini, Mauro Maccarrone, Marco Molinari

Endocannabinoids stimulate human melanogenesis via type-1 cannabinoid receptor

内源性大麻素通过 1 型大麻素受体刺激人类黑色素生成

Mariangela Pucci, Nicoletta Pasquariello, Natalia Battista, Monia Di Tommaso, Cinzia Rapino, Filomena Fezza, Michela Zuccolo, Roland Jourdain, Alessandro Finazzi Agrò, Lionel Breton, Mauro Maccarrone

Pitfalls and solutions in assaying anandamide transport in cells

检测细胞内花生四烯乙醇胺运输的陷阱和解决方案

Sergio Oddi, Filomena Fezza, Giuseppina Catanzaro, Chiara De Simone, Mariangela Pucci, Daniele Piomelli, Alessandro Finazzi-Agrò, Mauro Maccarrone