日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

BET inhibitor trotabresib in heavily pretreated patients with solid tumors and diffuse large B-cell lymphomas

BET 抑制剂 trotabresib 治疗接受过大量治疗的实体瘤和弥漫大 B 细胞淋巴瘤患者

Victor Moreno, Maria Vieito, Juan Manuel Sepulveda, Vladimir Galvao, Tatiana Hernández-Guerrero, Bernard Doger, Omar Saavedra, Carmelo Carlo-Stella, Jean-Marie Michot, Antoine Italiano, Massimo Magagnoli, Cecilia Carpio, Antonio Pinto, Rafael Sarmiento, Barbara Amoroso, Ida Aronchik, Ellen Filvaroff

Trotabresib, an oral potent bromodomain and extraterminal inhibitor, in patients with high-grade gliomas: A phase I, "window-of-opportunity" study

Trotabresib(一种口服强效溴结构域和末端结构域抑制剂)治疗高级别胶质瘤患者的 I 期“机会窗口”研究

Moreno, Victor; Manuel Sepúlveda, Juan; Reardon, David A; Pérez-Núñez, Ángel; González León, Pedro; Hanna, Bishoy; Filvaroff, Ellen; Aronchik, Ida; Chang, Henry; Amoroso, Barbara; Zuraek, Marlene; Sanchez-Perez, Tania; Mendez, Cristina; Stephens, Daniel; Nikolova, Zariana; Vogelbaum, Michael A

TACH101, a first-in-class pan-inhibitor of KDM4 histone demethylase

TACH101,首创的 KDM4 组蛋白去甲基化酶泛抑制剂

Chandtip Chandhasin, Van Dang, Frank Perabo, Joselyn Del Rosario, Young K Chen, Ellen Filvaroff, Jeffrey A Stafford, Michael Clarke

Trotabresib (CC-90010) in combination with adjuvant temozolomide or concomitant temozolomide plus radiotherapy in patients with newly diagnosed glioblastoma

Trotabresib (CC-90010) 联合辅助替莫唑胺或同步替莫唑胺加放疗用于新诊断的胶质母细胞瘤患者

Vieito, Maria; Simonelli, Matteo; de Vos, Filip; Moreno, Victor; Geurts, Marjolein; Lorenzi, Elena; Macchini, Marina; van den Bent, Martin J; Del Conte, Gianluca; de Jonge, Maja; Martín-Soberón, Maria Cruz; Amoroso, Barbara; Sanchez-Perez, Tania; Zuraek, Marlene; Hanna, Bishoy; Aronchik, Ida; Filvaroff, Ellen; Chang, Henry; Mendez, Cristina; Arias Parro, Marina; Wei, Xin; Nikolova, Zariana; Sepulveda, Juan Manuel

DNA-Dependent Protein Kinase Drives Prostate Cancer Progression through Transcriptional Regulation of the Wnt Signaling Pathway

DNA 依赖性蛋白激酶通过转录调控 Wnt 信号通路推动前列腺癌进展

Vishal Kothari, Jonathan F Goodwin, Shuang G Zhao, Justin M Drake, Yi Yin, S Laura Chang, Joseph R Evans, Kari Wilder-Romans, Kristina Gabbara, Emanuela Dylgjeri, Jonathan Chou, Grace Sun, Scott A Tomlins, Rohit Mehra, Kristen Hege, Ellen H Filvaroff, Edward M Schaeffer, R Jeffrey Karnes, David A Qu

First-In-Human Phase I Study Of A Dual mTOR Kinase And DNA-PK Inhibitor (CC-115) In Advanced Malignancy

针对晚期恶性肿瘤的双重 mTOR 激酶和 DNA-PK 抑制剂 (CC-115) 的首次人体 I 期研究

Munster, Pamela; Mita, Monica; Mahipal, Amit; Nemunaitis, John; Massard, Christophe; Mikkelsen, Tom; Cruz, Cristina; Paz-Ares, Luis; Hidalgo, Manuel; Rathkopf, Dana; Blumenschein, George Jr; Smith, David C; Eichhorst, Barbara; Cloughesy, Tim; Filvaroff, Ellen H; Li, Shaoyi; Raymon, Heather; de Haan, Hans; Hege, Kristen; Bendell, Johanna C

A technology platform to assess multiple cancer agents simultaneously within a patient's tumor

一种用于同时评估患者肿瘤内多种抗癌药物的技术平台

Klinghoffer, Richard A; Bahrami, S Bahram; Hatton, Beryl A; Frazier, Jason P; Moreno-Gonzalez, Alicia; Strand, Andrew D; Kerwin, William S; Casalini, Joseph R; Thirstrup, Derek J; You, Sheng; Morris, Shelli M; Watts, Korashon L; Veiseh, Mandana; Grenley, Marc O; Tretyak, Ilona; Dey, Joyoti; Carleton, Michael; Beirne, Emily; Pedro, Kyle D; Ditzler, Sally H; Girard, Emily J; Deckwerth, Thomas L; Bertout, Jessica A; Meleo, Karri A; Filvaroff, Ellen H; Chopra, Rajesh; Press, Oliver W; Olson, James M

MET Suppresses Epithelial VEGFR2 via Intracrine VEGF-induced Endoplasmic Reticulum-associated Degradation

MET 通过内分泌 VEGF 诱导的内质网相关降解抑制上皮 VEGFR2

Tom T Chen, Ellen Filvaroff, Jing Peng, Scot Marsters, Adrian Jubb, Hartmut Koeppen, Mark Merchant, Avi Ashkenazi

Biomarker analyses from a placebo-controlled phase II study evaluating erlotinib±onartuzumab in advanced non-small cell lung cancer: MET expression levels are predictive of patient benefit

一项评估厄洛替尼±奥那妥珠单抗治疗晚期非小细胞肺癌的安慰剂对照 II 期研究的生物标志物分析:MET 表达水平可预测患者获益

Hartmut Koeppen, Wei Yu, Jiping Zha, Ajay Pandita, Elicia Penuel, Linda Rangell, Rajiv Raja, Sankar Mohan, Rajesh Patel, Rupal Desai, Ling Fu, An Do, Vaishali Parab, Xiaoling Xia, Tom Januario, Sharianne G Louie, Ellen Filvaroff, David S Shames, Ignacio Wistuba, Marina Lipkind, Jenny Huang, Mirella

TGF-beta regulates the mechanical properties and composition of bone matrix

TGF-β调节骨基质的力学性能和组成

Balooch, Guive; Balooch, Mehdi; Nalla, Ravi K; Schilling, Stephen; Filvaroff, Ellen H; Marshall, Grayson W; Marshall, Sally J; Ritchie, Robert O; Derynck, Rik; Alliston, Tamara