日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Large Library Docking for Polypharmacology

用于多药理学的大型库对接

Wu, Yujin; Vigneron, Seth; Braz, Joao; Srinivasan, Karthik; Fink, Elissa A; Huang, Xi-Ping; Xu, Xinyu; Huebner, Harald; Kim, Joseph Y; Wang, Jing; Pfeiffer, Tara; Sakamoto, Kensuke; Radchenko, Dmytro S; Rodriguiz, Ramona M; Moroz, Yurii S; Irwin, John J; Gmeiner, Peter; Billesboelle, Christian; Roth, Bryan L; Basbaum, Allan I; Manglik, Aashish; Wetsel, William C; Shoichet, Brian K

Discovery of a functionally selective serotonin receptor (5-HT(1A)R) agonist for the treatment of pain.

发现一种功能选择性血清素受体(5-HT(1A)R)激动剂用于治疗疼痛

Ullrich Annika, Schneider Johannes, Braz João M, Neu Eduard, Staffen Nico, Stanek Markus, Bláhová Jana, Hove Tamsanqa, Albert Tamara, Allikalt Anni, Löber Stefan, Bhardwaj Karnika, Rodriguez-Rosado Sian, Fink Elissa, Rasmussen Tim, Hübner Harald, Inoue Asuka, Shoichet Brian K, Basbaum Allan I, Böttcher Bettina, Weikert Dorothee, Gmeiner Peter

A practical guide to large-scale docking

大规模对接实用指南

Bender, Brian J; Gahbauer, Stefan; Luttens, Andreas; Lyu, Jiankun; Webb, Chase M; Stein, Reed M; Fink, Elissa A; Balius, Trent E; Carlsson, Jens; Irwin, John J; Shoichet, Brian K

Robust Sequence Determinants of α-Synuclein Toxicity in Yeast Implicate Membrane Binding

酵母中α-突触核蛋白毒性的稳健序列决定因素表明其与膜结合有关

Newberry, Robert W; Arhar, Taylor; Costello, Jean; Hartoularos, George C; Maxwell, Alison M; Naing, Zun Zar Chi; Pittman, Maureen; Reddy, Nishith R; Schwarz, Daniel M C; Wassarman, Douglas R; Wu, Taia S; Barrero, Daniel; Caggiano, Christa; Catching, Adam; Cavazos, Taylor B; Estes, Laurel S; Faust, Bryan; Fink, Elissa A; Goldman, Miriam A; Gomez, Yessica K; Gordon, M Grace; Gunsalus, Laura M; Hoppe, Nick; Jaime-Garza, Maru; Johnson, Matthew C; Jones, Matthew G; Kung, Andrew F; Lopez, Kyle E; Lumpe, Jared; Martyn, Calla; McCarthy, Elizabeth E; Miller-Vedam, Lakshmi E; Navarro, Erik J; Palar, Aji; Pellegrino, Jenna; Saylor, Wren; Stephens, Christina A; Strickland, Jack; Torosyan, Hayarpi; Wankowicz, Stephanie A; Wong, Daniel R; Wong, Garrett; Redding, Sy; Chow, Eric D; DeGrado, William F; Kampmann, Martin