日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Extracting Mechanistic Information from an Open Data Set for a Pharma-Relevant Suzuki-Miyaura Cross-Coupling Reaction

从开放数据集中提取与制药相关的铃木-宫浦交叉偶联反应的机理信息

Franklin, Barnabas A; Donaldson, Niall W B; Firth, James D; Horbaczewskyj, Christopher S; Aspell, Aaron; Tanner, Theo; Whitwood, Adrian C; Wilson, Julie; Hargreaves, Jessica K; Fairlamb, Ian J S

Modular Synthetic Platform for the Elaboration of Fragments in Three Dimensions for Fragment-Based Drug Discovery

用于三维片段构建的模块化合成平台,以进行基于片段的药物发现

Gomez-Angel, Andres R; Klein, Hanna F; Yao, Stephen Y; Donald, James R; Firth, James D; Appiani, Rebecca; Palmer, Cameron J; Lincoln, Joshua; Lucas, Simon C C; Fusani, Lucia; Storer, R Ian; O'Brien, Peter

Design, modular synthesis and screening of 58 shape-diverse 3-D fragments

设计、模块化合成和筛选58种形状各异的三维片段

Downes, Thomas D; Jones, S Paul; Firth, James D; Darby, John F; Gilio, Amelia K; Klein, Hanna F; Wang, Xinyu; Blakemore, David C; De Fusco, Claudia; Roughley, Stephen D; Vidler, Lewis R; Whatton, Maria Ann; Woolford, Alison J-A; Wrigley, Gail L; Hubbard, Roderick E; Wu, Liang; Davies, Gideon J; O'Brien, Peter

α-Functionalisation of Cyclic Sulfides Enabled by Lithiation Trapping

锂化捕获实现环状硫化物的α-官能化

Seling, Nico; Atobe, Masakazu; Kasten, Kevin; Firth, James D; Karadakov, Peter B; Goldberg, Frederick W; O'Brien, Peter

Deciphering complexity in Pd-catalyzed cross-couplings

解读钯催化交叉偶联反应的复杂性

Clarke, George E; Firth, James D; Ledingham, Lyndsay A; Horbaczewskyj, Chris S; Bourne, Richard A; Bray, Joshua T W; Martin, Poppy L; Eastwood, Jonathan B; Campbell, Rebecca; Pagett, Alex; MacQuarrie, Duncan J; Slattery, John M; Lynam, Jason M; Whitwood, Adrian C; Milani, Jessica; Hart, Sam; Wilson, Julie; Fairlamb, Ian J S

Design and Synthesis of 56 Shape-Diverse 3D Fragments

设计并合成56种形状各异的三维碎片

Downes, Thomas D; Jones, S Paul; Klein, Hanna F; Wheldon, Mary C; Atobe, Masakazu; Bond, Paul S; Firth, James D; Chan, Ngai S; Waddelove, Laura; Hubbard, Roderick E; Blakemore, David C; De Fusco, Claudia; Roughley, Stephen D; Vidler, Lewis R; Whatton, Maria Ann; Woolford, Alison J-A; Wrigley, Gail L; O'Brien, Peter

Increase of enzyme activity through specific covalent modification with fragments

通过与片段进行特定的共价修饰来提高酶活性

Darby, John F; Atobe, Masakazu; Firth, James D; Bond, Paul; Davies, Gideon J; O'Brien, Peter; Hubbard, Roderick E

Lipopolysaccharide-induced epithelial monoamine oxidase mediates alveolar bone loss in a rat chronic wound model.

脂多糖诱导的上皮单胺氧化酶介导大鼠慢性伤口模型中的牙槽骨丢失

Ekuni Daisuke, Firth James D, Nayer Tarun, Tomofuji Takaaki, Sanbe Toshihiro, Irie Koichiro, Yamamoto Tatsuo, Oka Takashi, Liu Zhenzi, Vielkind Juergen, Putnins Edward E

Fusobacterium nucleatum increases collagenase 3 production and migration of epithelial cells

具核梭杆菌可增加胶原酶3的产生和上皮细胞的迁移。

Uitto, Veli-Jukka; Baillie, Daniel; Wu, Qiang; Gendron, Renee; Grenier, Daniel; Putnins, Edward E; Kanervo, Arja; Firth, James D