日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in Enterococcus faecium Septicemic Peritonitis Mouse Model While Sparing the Microbiome

细菌碳酸酐酶抑制剂 CAI0019 在粪肠球菌败血性腹膜炎小鼠模型中显示出疗效,同时不影响肠道菌群。

Abutaleb, Nader S; Holly, Katrina J; Metcalfe, Carolyn K; Abouelkhair, Ahmed A; Tharra, Prabhakara R; Shrinidhi, Annadka; Abdelsattar, Abdallah S; Burgo, Victoria; Melotte, Glory; Akin-Olabiyi, Tomi; Knoblauch, Sean; Ramaswamy, Ramanujam; Woodson, Che; Thirumalaikumar, Venkatesh P; Rodriguez, J Alejandra; Yeo, Franklin J; Snell, Olivia C; Nocentini, Alessio; Sundararajan, Anitha; Olson, Matthew R; Supuran, Claudiu T; Seleem, Mohamed N; Flaherty, Daniel P

Meet key digital health thought leaders: Sandy Engelhardt, Scientific Program Chair of the ESC’s Digital Summit 2025

与数字健康领域的重要思想领袖会面:桑迪·恩格尔哈特,ESC 2025数字峰会科学项目主席

Tang, Haiyang; Gupta, Akash; Morrisroe, Seth A; Bao, Changlei; Schwantes-An, Tae-Hwi; Gupta, Geetanjali; Liang, Shuxin; Sun, Yanan; Chu, Aiai; Luo, Ang; Ramamoorthi Elangovan, Venkateswaran; Sangam, Shreya; Shi, Yinan; Naidu, Samisubbu R; Jheng, Jia-Rong; Ciftci-Yilmaz, Sultan; Warfel, Noel A; Hecker, Louise; Mitra, Sumegha; Coleman, Anna W; Lutz, Katie A; Pauciulo, Michael W; Lai, Yen-Chun; Javaheri, Ali; Dharmakumar, Rohan; Wu, Wen-Hui; Flaherty, Daniel P; Karnes, Jason H; Breuils-Bonnet, Sandra; Boucherat, Olivier; Bonnet, Sebastien; Yuan, Jason X-J; Jacobson, Jeffrey R; Duarte, Julio D; Nichols, William C; Garcia, Joe G N; Desai, Ankit A; Bruining, Nico

Hit-to-Lead Optimization of Acetazolamide-Based Bacterial Carbonic Anhydrase Inhibitors with Efficacy In Vivo for Treatment of Vancomycin-Resistant Enterococci Septicemia

基于乙酰唑胺的细菌碳酸酐酶抑制剂的先导化合物优化,以评估其在体内治疗耐万古霉素肠球菌败血症的疗效。

Holly, Katrina J; Tharra, Prabhakara R; Abutaleb, Nader S; Nocentini, Alessio; Abouelkhair, Ahmed A; Youse, Molly S; Marapaka, Anil Kumar; S Abdelsattar, Abdallah; An, Weiwei; Drummond, Faith L; Snell, Olivia C; Supuran, Claudiu T; Seleem, Mohamed N; Flaherty, Daniel P

Optimization of Ethoxzolamide Analogs with Improved Pharmacokinetic Properties for In Vivo Efficacy against Neisseria gonorrhoeae.

优化乙氧唑胺类似物,提高其药代动力学特性,以增强其对淋病奈瑟菌的体内疗效

Youse Molly S, Abutaleb Nader S, Nocentini Alessio, S Abdelsattar Abdallah, Ali Farman, Supuran Claudiu T, Seleem Mohamed N, Flaherty Daniel P

Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae.

针对耐多药淋病奈瑟菌的青霉素类碳酸酐酶抑制剂的研发

Bonardi Alessandro, Nocentini Alessio, Giovannuzzi Simone, Paoletti Niccolò, Ammara Andrea, Bua Silvia, Abutaleb Nader S, Abdelsattar Abdallah S, Capasso Clemente, Gratteri Paola, Flaherty Daniel P, Seleem Mohamed N, Supuran Claudiu T

Biochemical pharmacology of adenylyl cyclases in cancer

癌症中腺苷酸环化酶的生化药理学

Chandra Jena, Bikash; Flaherty, Daniel P; O'Brien, Valerie P; Watts, Val J

Unguarded liabilities: Borrelia burgdorferi's complex amino acid dependence exposes unique avenues of inhibition

未被防范的风险:伯氏疏螺旋体复杂的氨基酸依赖性暴露出独特的抑制途径

Holly, Katrina J; Kataria, Arti; Flaherty, Daniel P; Groshong, Ashley M

Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates

单硫代氨基甲酸酯对致病菌碳酸酐酶的抑制作用

Giovannuzzi, Simone; Marapaka, Anil Kumar; Abutaleb, Nader S; Carta, Fabrizio; Liang, Hsin-Wen; Nocentini, Alessio; Pisano, Luigi; Seleem, Mohamed N; Flaherty, Daniel P; Supuran, Claudiu T

Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to Neisseria gonorrhoeae α-Carbonic Anhydrase

噻二唑磺酰胺类抑制剂与淋病奈瑟菌α-碳酸酐酶结合的结构表征

Marapaka, Anil Kumar; Nocentini, Alessio; Youse, Molly S; An, Weiwei; Holly, Katrina J; Das, Chittaranjan; Yadav, Ravi; Seleem, Mohamed N; Supuran, Claudiu T; Flaherty, Daniel P

Evaluation of 1,3,4-Thiadiazole Carbonic Anhydrase Inhibitors for Gut Decolonization of Vancomycin-Resistant Enterococci

评价 1,3,4-噻二唑碳酸酐酶抑制剂对肠道中耐万古霉素肠球菌的清除作用

Abutaleb, Nader S; Shrinidhi, Annadka; Bandara, Aloka B; Seleem, Mohamed N; Flaherty, Daniel P