Synthesis of bis-furyl-pyrrolo[3,4-b]pyridin-5-ones via Ugi-Zhu reaction and in vitro activity assays against human SARS-CoV-2 and in silico studies on its main proteins.
通过 Ugi-Zhu 反应合成双呋喃基吡咯并[3,4-b]吡啶-5-酮,并进行针对人类 SARS-CoV-2 的体外活性测定和对其主要蛋白质的计算机模拟研究
期刊:RSC Medicinal Chemistry
影响因子:3.6
doi:10.1039/d2md00350c
Morales-Salazar Ivette, Montes-EnrÃquez Flora P, Garduño-Albino Carlos E, GarcÃa-Sánchez M A, Ibarra Ilich A, Rojas-Aguirre Yareli, GarcÃa-Hernández Montserrat Elemi, Sarmiento-Silva Rosa Elena, Alcaraz-Estrada SofÃa Lizeth, DÃaz-Cervantes Erik, González-Zamora Eduardo, Islas-Jácome Alejandro