Discovery of the First Selective M(4) Muscarinic Acetylcholine Receptor Antagonists with in Vivo Antiparkinsonian and Antidystonic Efficacy
发现首个具有体内抗帕金森病和抗肌张力障碍疗效的选择性M(4)毒蕈碱乙酰胆碱受体拮抗剂
期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.0c00162
Moehle, Mark S; Bender, Aaron M; Dickerson, Jonathan W; Foster, Daniel J; Qi, Aidong; Cho, Hyekyung P; Donsante, Yuping; Peng, Weimin; Bryant, Zoey; Stillwell, Kaylee J; Bridges, Thomas M; Chang, Sichen; Watson, Katherine J; O'Neill, Jordan C; Engers, Julie L; Peng, Li; Rodriguez, Alice L; Niswender, Colleen M; Lindsley, Craig W; Hess, Ellen J; Conn, P Jeffrey; Rook, Jerri M