日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Thioquinazolinones as Antituberculosis Agents Targeting Phosphopantetheinyl Transferase

硫代喹唑啉酮类化合物作为靶向磷酸泛酰巯基转移酶的抗结核药物

Singh, Amrita; Zwerneman, Logan T; Planck, Kyle; Kaneko, Takushi; Perkowski, Andrew J; Suh, Christine M; Alex, Alexander; Bean, James; Burns-Huang, Kristin; Zhang, David; Boshoff, Helena I M; Roubert, Christine; Krieger, Inna; Gardner, Mark; Cautain, Bastien; Cooper, Christopher B; Tanvir, Zaid; Sacchettini, James; Gold, Ben S; Rhee, Kyu Y; Fotouhi, Nader; Nathan, Carl F; Aubé, Jeffrey

Contribution of telacebec to novel drug regimens in a murine tuberculosis model

替拉西贝克对小鼠结核病模型中新型药物治疗方案的贡献

Komm, Oliver D; Tyagi, Sandeep; Garcia, Andrew; Almeida, Deepak; Chang, Yong; Li, Si-Yang; Castillo, Jennie Ruelas; Converse, Paul J; Black, Todd; Fotouhi, Nader; Nuermberger, Eric L

Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase.

将 raltitrexed 从癌细胞胸苷酸合成酶重定向到结核分枝杆菌磷酸泛酰巯基转移酶

Singh Amrita, Ottavi Samantha, Krieger Inna, Planck Kyle, Perkowski Andrew, Kaneko Takushi, Davis Andrew M, Suh Christine, Zhang David, Goullieux Laurent, Alex Alexander, Roubert Christine, Gardner Mark, Preston Marian, Smith Dave M, Ling Yan, Roberts Julia, Cautain Bastien, Upton Anna, Cooper Christopher B, Serbina Natalya, Tanvir Zaid, Mosior John, Ouerfelli Ouathek, Yang Guangli, Gold Ben S, Rhee Kyu Y, Sacchettini James C, Fotouhi Nader, Aubé Jeffrey, Nathan Carl

Relative Contributions of the Novel Diarylquinoline TBAJ-876 and its Active Metabolite to the Bactericidal Activity in a Murine Model of Tuberculosis

新型二芳基喹啉类化合物TBAJ-876及其活性代谢物在小鼠结核病模型中杀菌活性的相对贡献

Mudde, Saskia E; Ammerman, Nicole C; Ten Kate, Marian T; Fotouhi, Nader; Lotlikar, Manisha U; Bax, Hannelore I; de Steenwinkel, Jurriaan E M

Bactericidal and sterilizing activity of novel regimens combining bedaquiline or TBAJ-587 with GSK2556286 and TBA-7371 in a mouse model of tuberculosis

在结核病小鼠模型中,贝达喹啉或TBAJ-587与GSK2556286和TBA-7371联合使用的新方案的杀菌和灭菌活性

Li, Si-Yang; Tyagi, Sandeep; Soni, Heena; Betoudji, Fabrice; Converse, Paul J; Mdluli, Khisimuzi; Upton, Anna M; Fotouhi, Nader; Barros-Aguirre, David; Ballell, Lluís; Jimenez-Navarro, Elena; Nuermberger, Eric L

Contribution of direct InhA inhibitors to novel drug regimens in a mouse model of tuberculosis

直接InhA抑制剂对结核病小鼠模型新型药物治疗方案的贡献

Encinas, Lourdes; Li, Si-Yang; Rullas-Trincado, Joaquin; Tasneen, Rokeya; Tyagi, Sandeep; Soni, Heena; Garcia-Perez, Adolfo; Lee, Jin; González Del Río, Rubén; De Mercado, Jaime; Sousa, Verónica; Sosič, Izidor; Gobec, Stanislav; Mendoza-Losana, Alfonso; Converse, Paul J; Mdluli, Khisi; Fotouhi, Nader; Barros-Aguirre, David; Nuermberger, Eric L

Combating antimicrobial resistance in malaria, HIV and tuberculosis

对抗疟疾、艾滋病和结核病中的抗菌素耐药性

Duffey, Maëlle; Shafer, Robert W; Timm, Juliano; Burrows, Jeremy N; Fotouhi, Nader; Cockett, Mark; Leroy, Didier

Next-Generation Diarylquinolines Improve Sterilizing Activity of Regimens with Pretomanid and the Novel Oxazolidinone TBI-223 in a Mouse Tuberculosis Model

在小鼠结核病模型中,新一代二芳基喹啉类化合物可提高普瑞托马尼和新型噁唑烷酮类药物TBI-223联合治疗方案的杀菌活性。

Li, Si-Yang; Converse, Paul J; Betoudji, Fabrice; Lee, Jin; Mdluli, Khisimuzi; Upton, Anna; Fotouhi, Nader; Nuermberger, Eric L

Contezolid can replace linezolid in a novel combination with bedaquiline and pretomanid in a murine model of tuberculosis

在结核病小鼠模型中,康替唑利德可以替代利奈唑胺,与贝达喹啉和普瑞托马尼联合使用。

Almeida, Deepak; Li, Si-Yang; Lee, Jin; Hafkin, Barry; Mdluli, Khisimuzi; Fotouhi, Nader; Nuermberger, Eric L

Identification of 2-Aryl-Quinolone Inhibitors of Cytochrome bd and Chemical Validation of Combination Strategies for Respiratory Inhibitors against Mycobacterium tuberculosis

鉴定细胞色素bd的2-芳基喹诺酮抑制剂及抗结核分枝杆菌呼吸抑制剂组合策略的化学验证

Jeffreys, Laura N; Ardrey, Alison; Hafiz, Taghreed A; Dyer, Lauri-Anne; Warman, Ashley J; Mosallam, Nada; Nixon, Gemma L; Fisher, Nicholas E; Hong, W David; Leung, Suet C; Aljayyoussi, Ghaith; Bibby, Jaclyn; Almeida, Deepak V; Converse, Paul J; Fotouhi, Nader; Berry, Neil G; Nuermberger, Eric L; Upton, Anna M; O'Neill, Paul M; Ward, Stephen A; Biagini, Giancarlo A