日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Highly Potent Small Molecule Pan-Coronavirus Fusion Inhibitors

发现高效小分子泛冠状病毒融合抑制剂

Francesca Curreli, Kent Chau, Thanh-Thuy Tran, Isabella Nicolau, Shahad Ahmed, Pujita Das, Christopher D Hillyer, Mary Premenko-Lanier, Asim K Debnath

Discovery of Highly Potent Fusion Inhibitors with Potential Pan-Coronavirus Activity That Effectively Inhibit Major COVID-19 Variants of Concern (VOCs) in Pseudovirus-Based Assays

发现具有潜在泛冠状病毒活性的高效融合抑制剂,可在基于假病毒的检测中有效抑制主要 COVID-19 变异株 (VOC)

Francesca Curreli, Shahad Ahmed, Sofia M B Victor, Aleksandra Drelich, Siva S Panda, Andrea Altieri, Alexander V Kurkin, Chien-Te K Tseng, Christopher D Hillyer, Asim K Debnath

Stapled Peptides Based on Human Angiotensin-Converting Enzyme 2 (ACE2) Potently Inhibit SARS-CoV-2 Infection In Vitro

基于人类血管紧张素转换酶 2 (ACE2) 的钉合肽在体外有效抑制 SARS-CoV-2 感染

Francesca Curreli, Sofia M B Victor, Shahad Ahmed, Aleksandra Drelich, Xiaohe Tong, Chien-Te K Tseng, Christopher D Hillyer, Asim K Debnath

Identification of Combinations of Protein Kinase C Activators and Histone Deacetylase Inhibitors That Potently Reactivate Latent HIV

鉴定可有效重新激活潜伏 HIV 的蛋白激酶 C 激活剂和组蛋白去乙酰化酶抑制剂的组合

Francesca Curreli, Shahad Ahmed, Sofia M Benedict Victor, Asim K Debnath

Blood Cell-Bound C4d as a Marker of Complement Activation in Patients With the Antiphospholipid Syndrome

抗磷脂综合征患者血细胞结合C4d作为补体激活的标志物

Lonati, Paola Adele; Scavone, Mariangela; Gerosa, Maria; Borghi, Maria Orietta; Pregnolato, Francesca; Curreli, Daniele; Podda, Gianmarco; Femia, Eti Alessandra; Barcellini, Wilma; Cattaneo, Marco; Tedesco, Francesco; Meroni, Pier Luigi

Structure-based lead optimization to improve antiviral potency and ADMET properties of phenyl-1H-pyrrole-carboxamide entry inhibitors targeted to HIV-1 gp120

基于结构的先导优化可提高针对 HIV-1 gp120 的苯基-1H-吡咯-酰胺进入抑制剂的抗病毒效力和 ADMET 特性

Francesca Curreli, Dmitry S Belov, Young Do Kwon, Ranjith Ramesh, Anna M Furimsky, Kathleen O'Loughlin, Patricia C Byrge, Lalitha V Iyer, Jon C Mirsalis, Alexander V Kurkin, Andrea Altieri, Asim K Debnath

Anti-inflammatory effects of H(2)S during acute bacterial infection: a review

H₂S在急性细菌感染中的抗炎作用:综述

Benedetti, Francesca; Curreli, Sabrina; Krishnan, Selvi; Davinelli, Sergio; Cocchi, Fiorenza; Scapagnini, Giovanni; Gallo, Robert C; Zella, Davide

Structure-Based Design of a Small Molecule CD4-Antagonist with Broad Spectrum Anti-HIV-1 Activity

基于结构的设计具有广谱抗 HIV-1 活性的小分子 CD4 拮抗剂

Francesca Curreli #, Young Do Kwon #, Hongtao Zhang, Daniel Scacalossi, Dmitry S Belov, Artur A Tikhonov, Ivan A Andreev, Andrea Altieri, Alexander V Kurkin, Peter D Kwong, Asim K Debnath

Binding mode characterization of NBD series CD4-mimetic HIV-1 entry inhibitors by X-ray structure and resistance study

通过 X 射线结构和抗性研究对 NBD 系列 CD4 类似物 HIV-1 进入抑制剂的结合模式进行表征

Francesca Curreli, Young Do Kwon, Hongtao Zhang, Yongping Yang, Daniel Scacalossi, Peter D Kwong, Asim K Debnath

Dual-acting stapled peptides target both HIV-1 entry and assembly

双重作用的钉合肽靶向 HIV-1 进入和组装

Hongtao Zhang, Francesca Curreli, Abdul A Waheed, Peter Y Mercredi, Mansi Mehta, Pallavi Bhargava, Daniel Scacalossi, Xiaohe Tong, Shawn Lee, Alan Cooper, Michael F Summers, Eric O Freed, Asim K Debnath