日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Non-covalent inhibitors of thioredoxin glutathione reductase with schistosomicidal activity in vivo

具有体内杀血吸虫活性的硫氧还蛋白谷胱甘肽还原酶非共价抑制剂

Valentina Z Petukhova #, Sammy Y Aboagye #, Matteo Ardini #, Rachel P Lullo, Francesca Fata, Margaret E Byrne, Federica Gabriele, Lucy M Martin, Luke N M Harding, Vamshikrishna Gone, Bikash Dangi, Daniel D Lantvit, Dejan Nikolic, Rodolfo Ippoliti, Grégory Effantin, Wai Li Ling, Jeremy J Johnson, Gre

Biochemical and structural characterizations of thioredoxin reductase selenoproteins of the parasitic filarial nematodes Brugia malayi and Onchocerca volvulus

寄生丝虫马来丝虫和盘尾丝虫的硫氧还蛋白还原酶硒蛋白的生化和结构特征

Francesca Fata, Radosveta Gencheva, Qing Cheng, Rachel Lullo, Matteo Ardini, Ilaria Silvestri, Federica Gabriele, Rodolfo Ippoliti, Christina A Bulman, Judy A Sakanari, David L Williams, Elias S J Arnér, Francesco Angelucci

Probing the Surface of a Parasite Drug Target Thioredoxin Glutathione Reductase Using Small Molecule Fragments

利用小分子片段探测寄生虫药物靶标硫氧还蛋白谷胱甘肽还原酶的表面

Francesca Fata, Ilaria Silvestri, Matteo Ardini, Rodolfo Ippoliti, Luana Di Leandro, Nicola Demitri, Maurizio Polentarutti, Adele Di Matteo, Haining Lyu, Gregory R J Thatcher, Pavel A Petukhov, David L Williams, Francesco Angelucci

Ectopic suicide inhibition of thioredoxin glutathione reductase

异位自杀抑制硫氧还蛋白谷胱甘肽还原酶

Ilaria Silvestri, Haining Lyu, Francesca Fata, Paul R Banta, Benedetta Mattei, Rodolfo Ippoliti, Andrea Bellelli, Giuseppina Pitari, Matteo Ardini, Valentina Petukhova, Gregory R J Thatcher, Pavel A Petukhov, David L Williams, Francesco Angelucci

Fragment-Based Discovery of a Regulatory Site in Thioredoxin Glutathione Reductase Acting as "Doorstop" for NADPH Entry

基于片段的硫氧还蛋白谷胱甘肽还原酶中调节位点的发现,该位点充当 NADPH 进入的“门挡”

Ilaria Silvestri, Haining Lyu, Francesca Fata, Giovanna Boumis, Adriana E Miele, Matteo Ardini, Rodolfo Ippoliti, Andrea Bellelli, Ajit Jadhav, Wendy A Lea, Anton Simeonov, Qing Cheng, Elias S J Arnér, Gregory R J Thatcher, Pavel A Petukhov, David L Williams, Francesco Angelucci