日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural basis for the ligand-dependent activation of heterodimeric AHR-ARNT complex

异二聚体 AHR-ARNT 复合物的配体依赖性活化的结构基础

Xiaotong Diao #, Qinghong Shang #, Mengqi Guo, Yubin Huang, Meina Zhang, Xiaoyu Chen, Yinping Liang, Xiangnan Sun, Fan Zhou, Jingjing Zhuang, Shuang-Jiang Liu, Christoph F A Vogel, Fraydoon Rastinejad, Dalei Wu

Pharmacological targeting of BMAL1 modulates circadian and immune pathways

BMAL1的药理学靶向作用调节昼夜节律和免疫通路

Hua Pu ,Laura C Bailey ,Ludwig G Bauer ,Maria Voronkov ,Matthew Baxter ,Kilian V M Huber ,Sepideh Khorasanizadeh ,David Ray ,Fraydoon Rastinejad

Monoterpenoid aryl hydrocarbon receptor allosteric antagonists protect against ultraviolet skin damage in female mice

单萜芳烃受体变构拮抗剂可保护雌性小鼠免受紫外线皮肤损伤

Karolína Ondrová, Iveta Zůvalová, Barbora Vyhlídalová, Kristýna Krasulová, Eva Miková, Radim Vrzal, Petr Nádvorník, Binod Nepal, Sandhya Kortagere, Martina Kopečná, David Kopečný, Marek Šebela, Fraydoon Rastinejad, Hua Pu, Miroslav Soural, Katharina Maria Rolfes, Thomas Haarmann-Stemmann, Hao Li, Sr

The protein architecture and allosteric landscape of HNF4α

HNF4α的蛋白质结构和变构特性

Rastinejad, Fraydoon

Human gut bacteria produce ΤΗ17-modulating bile acid metabolites

人类肠道细菌产生调节TH17的胆汁酸代谢物

Donggi Paik # ,Lina Yao # ,Yancong Zhang ,Sena Bae ,Gabriel D D'Agostino ,Minghao Zhang ,Eunha Kim ,Eric A Franzosa ,Julian Avila-Pacheco ,Jordan E Bisanz ,Christopher K Rakowski ,Hera Vlamakis ,Ramnik J Xavier ,Peter J Turnbaugh ,Randy S Longman ,Michael R Krout ,Clary B Clish ,Fraydoon Rastinejad ,Curtis Huttenhower ,Jun R Huh ,A Sloan Devlin

Identification of oleoylethanolamide as an endogenous ligand for HIF-3α

油酰乙醇酰胺作为 HIF-3α 内源性配体的鉴定

Xiaotong Diao #, Fei Ye #, Meina Zhang, Xintong Ren, Xiaoxu Tian, Jingping Lu, Xiangnan Sun, Zeng Hou, Xiaoyu Chen, Fengwei Li, Jingjing Zhuang, Hong Ding, Chao Peng, Fraydoon Rastinejad, Cheng Luo, Dalei Wu

The Highly Potent AhR Agonist Picoberin Modulates Hh-Dependent Osteoblast Differentiation

高效 AhR 激动剂 Picoberin 调节 Hh 依赖性成骨细胞分化

Jana Flegel, Saad Shaaban, Zhi Jun Jia, Britta Schulte, Yilong Lian, Adrian Krzyzanowski, Malte Metz, Tabea Schneidewind, Fabian Wesseler, Anke Flegel, Alisa Reich, Alexandra Brause, Gang Xue, Minghao Zhang, Lara Dötsch, Isabelle D Stender, Jan-Erik Hoffmann, Rebecca Scheel, Petra Janning, Fraydoon

Retinoic acid receptor structures: the journey from single domains to full-length complex

视黄酸受体结构:从单个结构域到全长复合物的演变

Rastinejad, Fraydoon

Structures of NPAS4-ARNT and NPAS4-ARNT2 heterodimers reveal new dimerization modalities in the bHLH-PAS transcription factor family

NPAS4-ARNT 和 NPAS4-ARNT2 异二聚体的结构揭示了 bHLH-PAS 转录因子家族中的新二聚化方式

Xiangnan Sun, Linqian Jing, Fengwei Li, Meina Zhang, Xiaotong Diao, Jingjing Zhuang, Fraydoon Rastinejad, Dalei Wu

A bacterial bile acid metabolite modulates Treg activity through the nuclear hormone receptor NR4A1

细菌胆汁酸代谢产物通过核激素受体NR4A1调节Treg细胞活性

Wei Li ,Saiyu Hang ,Yuan Fang ,Sena Bae ,Yancong Zhang ,Minghao Zhang ,Gang Wang ,Megan D McCurry ,Munhyung Bae ,Donggi Paik ,Eric A Franzosa ,Fraydoon Rastinejad ,Curtis Huttenhower ,Lina Yao ,A Sloan Devlin ,Jun R Huh