日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Naphthalene diimide-naphthalimide dyads promote telomere damage by selectively targeting multimeric G-quadruplexes.

萘二酰亚胺-萘酰亚胺二聚体通过选择性靶向多聚体 G-四链体促进端粒损伤

Pirota Valentina, Iachettini Sara, Platella Chiara, Zizza Pasquale, Fracchioni Giorgia, Di Vito Serena, Carachino Alice, Battistini Federica, Orozco Modesto, Freccero Mauro, Biroccio Annamaria, Montesarchio Daniela, Doria Filippo

Core-Extended Naphthalene Diimide Dyads as Light-Up Probes with Targeted Cytotoxicity Toward Tumor Cells

核心延伸的萘二酰亚胺二聚体作为对肿瘤细胞具有靶向细胞毒性的光敏探针

Pirota, Valentina; Salvati, Erica; Risoldi, Carla; Manoli, Francesco; Rizzo, Angela; Zizza, Pasquale; Biroccio, Annamaria; Freccero, Mauro; Manet, Ilse; Doria, Filippo

A Novel G-Quadruplex Structure within Apolipoprotein E Promoter: A New Promising Target in Cancer and Dementia Fight?

载脂蛋白E启动子中一种新型G-四链体结构:癌症和痴呆症治疗中一个有前景的新靶点?

Pirota, Valentina; Stritto, Angela Dello; Magnaghi, Lisa Rita; Biesuz, Raffaela; Doria, Filippo; Mella, Mariella; Freccero, Mauro; Crespan, Emmanuele

Naphthalene Diimide-Tetraazacycloalkane Conjugates Are G-Quadruplex-Based HIV-1 Inhibitors with a Dual Mode of Action

萘二酰亚胺-四氮杂环烷烃缀合物是基于G-四链体的HIV-1抑制剂,具有双重作用机制

Nadai, Matteo; Doria, Filippo; Frasson, Ilaria; Perrone, Rosalba; Pirota, Valentina; Bergamaschi, Greta; Freccero, Mauro; Richter, Sara N

Studying the Dynamics of a Complex G-Quadruplex System: Insights into the Comparison of MD and NMR Data

研究复杂G-四链体系统的动力学:MD和NMR数据比较的启示

Castelli, Matteo; Doria, Filippo; Freccero, Mauro; Colombo, Giorgio; Moroni, Elisabetta

Selective Recognition of a Single HIV-1 G-Quadruplex by Ultrafast Small-Molecule Screening

利用超快速小分子筛选技术选择性识别单个 HIV-1 G-四链体

Scalabrin, Matteo; Nadai, Matteo; Tassinari, Martina; Lago, Sara; Doria, Filippo; Frasson, Ilaria; Freccero, Mauro; Richter, Sara N

Selective Binding and Redox-Activity on Parallel G-Quadruplexes by Pegylated Naphthalene Diimide-Copper Complexes

聚乙二醇化萘二酰亚胺-铜配合物对平行G-四链体的选择性结合和氧化还原活性

Pirota, Valentina; Lunghi, Enrico; Benassi, Alessandra; Crespan, Emmanuele; Freccero, Mauro; Doria, Filippo

New perspectives in cancer drug development: computational advances with an eye to design

癌症药物研发的新视角:着眼于设计的计算进展

Castelli, Matteo; Serapian, Stefano A; Marchetti, Filippo; Triveri, Alice; Pirota, Valentina; Torielli, Luca; Collina, Simona; Doria, Filippo; Freccero, Mauro; Colombo, Giorgio

Selective targeting of mutually exclusive DNA G-quadruplexes: HIV-1 LTR as paradigmatic model

选择性靶向互斥的DNA G-四链体:以HIV-1 LTR为例

Tassinari, Martina; Zuffo, Michela; Nadai, Matteo; Pirota, Valentina; Sevilla Montalvo, Adriana Carolina; Doria, Filippo; Freccero, Mauro; Richter, Sara N

On the interaction of an anticancer trisubstituted naphthalene diimide with G-quadruplexes of different topologies: a structural insight

抗癌三取代萘二酰亚胺与不同拓扑结构的G-四链体相互作用的结构解析

Platella, Chiara; Trajkovski, Marko; Doria, Filippo; Freccero, Mauro; Plavec, Janez; Montesarchio, Daniela