Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric Modulator
发现MK-8768,一种强效且选择性的mGluR2负变构调节剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.3c00210
Rudd, Michael T; Manley, Peter J; Hanney, Barbara; Meng, Zhaoyang; Shu, Youheng; de Leon, Pablo; Frie, Jessica L; Han, Yongxin; Wai, Jenny Miu-Chun; Yang, Zhi-Qiang; Perkins, James J; Hurzy, Danielle M; Manikowski, Jesse J; Zhu, Hong; Bungard, Christopher J; Converso, Antonella; Meissner, Robert S; Cosden, Mali L; Hayashi, Ikuo; Ma, Lei; O'Brien, Julie; Uebele, Victor N; Schachter, Joel B; Bhandari, Neetesh; Ward, Gwendolyn J; Fillgrove, Kerry L; Lu, Bing; Liang, Yuexia; Dubost, David C; Puri, Vanita; Eddins, Donnie M; Vardigan, Joshua D; Drolet, Robert E; Kern, Jonathan T; Uslaner, Jason M