日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

From Pharmacophore to Warhead: NAD(+)-Targeting Triazoles as Mechanism-Based Sirtuin Inhibitors

从药效团到活性位点:靶向 NAD(+) 的三唑类化合物作为基于机制的 Sirtuin 抑制剂

Friedrich, Florian; Meleshin, Marat; Papenkordt, Niklas; Gaitzsch, Lena; Prucker, Isabel; Borso, Marco; Ruprecht, Jan; Vorreiter, Christopher; Rast, Sabrina; Zhang, Lin; Schiedel, Matthias; Sippl, Wolfgang; Imhof, Axel; Jessen, Henning J; Einsle, Oliver; Schutkowski, Mike; Jung, Manfred

Molecular determinants for recognition of serotonylated chromatin

识别血清素化染色质的分子决定因素

Pulido-Cortés, Laura; Gielingh, Hajo; Thijssen, Vito; Liu, Minglong; Yoshisada, Ryoji; Romão Soares, Leonardo; Nizamuddin, Sheikh; Friedrich, Florian; Greschik, Holger; Peng, Ling; Vargas Honorato, Rodrigo; Jung, Manfred; Bonvin, Alexandre M J J; Biniossek, Martin L; Schüle, Roland; Jongkees, Seino; van Ingen, Hugo; Timmers, H Th Marc

Efficient Crystallization of Apo Sirt2 for Small-Molecule Soaking and Structural Analysis of Ligand Interactions.

高效结晶 Apo Sirt2 用于小分子浸泡和配体相互作用的结构分析

Friedrich Florian, Schiedel Matthias, Swyter Sören, Zhang Lin, Sippl Wolfgang, Schutkowski Mike, Einsle Oliver, Jung Manfred

Tailored SirReal-type inhibitors enhance SIRT2 inhibition through ligand stabilization and disruption of NAD(+) co-factor binding.

定制的 SirReal 型抑制剂通过配体稳定和破坏 NAD(+) 辅因子结合来增强 SIRT2 抑制作用

Wirawan Ricky, Frei Matthias, Heider Anna, Papenkordt Niklas, Friedrich Florian, Wein Thomas, Jung Manfred, Groll Michael, Huber Eva M, Bracher Franz

Structural Insights into Broad-Range Polyphosphate Kinase 2-II Enzymes Applicable for Pyrimidine Nucleoside Diphosphate Synthesis

广谱多聚磷酸激酶2-II酶的结构解析及其在嘧啶核苷二磷酸合成中的应用

Kuge, Marco; Keppler, Michael; Friedrich, Florian; Saleem-Batcha, Raspudin; Winter, Juliana; Prucker, Isabel; Germer, Philipp; Gerhardt, Stefan; Einsle, Oliver; Jung, Manfred; Jessen, Henning J; Andexer, Jennifer N

Beyond T2 and 3T: New MRI techniques for clinicians

超越T2和3T:面向临床医生的新型MRI技术

Knowles, Benjamin R; Friedrich, Florian; Fischer, Carola; Paech, Daniel; Ladd, Mark E

Cell-Cycle Position of Single MYC-Driven Cancer Cells Dictates Their Susceptibility to a Chemotherapeutic Drug

单个 MYC 驱动的癌细胞的细胞周期位置决定了它们对化疗药物的敏感性

Tatsiana Ryl, Erika E Kuchen, Emma Bell, Chunxuan Shao, Andrés F Flórez, Gregor Mönke, Sina Gogolin, Mona Friedrich, Florian Lamprecht, Frank Westermann, Thomas Höfer

Raman difference spectroscopy: a non-invasive method for identification of oral squamous cell carcinoma

拉曼差分光谱法:一种用于识别口腔鳞状细胞癌的非侵入性方法

Christian, Knipfer; Johanna, Motz; Werner, Adler; Kathrin, Brunner; Tesfay, Gebrekidan Medhaine; Robert, Hankel; Abbas, Agaimy; Stefan, Will; Andreas, Braeuer; Wilhelm, Neukam Friedrich; Florian, Stelzle