From Pharmacophore to Warhead: NAD(+)-Targeting Triazoles as Mechanism-Based Sirtuin Inhibitors
从药效团到活性位点:靶向 NAD(+) 的三唑类化合物作为基于机制的 Sirtuin 抑制剂
期刊:Angewandte Chemie-International Edition
影响因子:16.9
doi:10.1002/anie.202516782
Friedrich, Florian; Meleshin, Marat; Papenkordt, Niklas; Gaitzsch, Lena; Prucker, Isabel; Borso, Marco; Ruprecht, Jan; Vorreiter, Christopher; Rast, Sabrina; Zhang, Lin; Schiedel, Matthias; Sippl, Wolfgang; Imhof, Axel; Jessen, Henning J; Einsle, Oliver; Schutkowski, Mike; Jung, Manfred