日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Achieving well-informed decision-making in drug discovery: a comprehensive calibration study using neural network-based structure-activity models

在药物发现中实现明智的决策:基于神经网络的构效关系模型的综合校准研究

Friesacher, Hannah Rosa; Engkvist, Ola; Mervin, Lewis; Moreau, Yves; Arany, Adam

β subunits of GABAA receptors form proton-gated chloride channels: Insights into the molecular basis

GABAA 受体 β 亚基形成质子门控氯离子通道:深入了解其分子基础

Aleksandra Garifulina, Theres Friesacher, Marco Stadler, Eva-Maria Zangerl-Plessl, Margot Ernst, Anna Stary-Weinzinger, Anita Willam, Steffen Hering

A selectivity filter mutation provides insights into gating regulation of a K(+) channel

选择性过滤器突变为钾离子通道的门控调控提供了新的见解

Friesacher, Theres; Reddy, Haritha P; Bernsteiner, Harald; Carlo Combista, J; Shalomov, Boris; Bera, Amal K; Zangerl-Plessl, Eva-Maria; Dascal, Nathan; Stary-Weinzinger, Anna

Development of IKATP Ion Channel Blockers Targeting Sulfonylurea Resistant Mutant KIR6.2 Based Channels for Treating DEND Syndrome

开发针对磺酰脲类药物耐药突变型 KIR6.2 通道的 IKATP 离子通道阻滞剂用于治疗 DEND 综合征

Marien J C Houtman, Theres Friesacher, Xingyu Chen, Eva-Maria Zangerl-Plessl, Marcel A G van der Heyden, Anna Stary-Weinzinger

RNA polymerase II-binding aptamers in human ACRO1 satellites disrupt transcription in cis

人类 ACRO1 卫星中的 RNA 聚合酶 II 结合适体破坏顺式转录

Jennifer L Boots, Frederike von Pelchrzim, Adam Weiss, Bob Zimmermann, Theres Friesacher, Maximilian Radtke, Marek Żywicki, Doris Chen, Katarzyna Matylla-Kulińska, Bojan Zagrovic, Renée Schroeder