日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Insights into PCSK9-LDLR Regulation and Trafficking via the Differential Functions of MHC-I Proteins HFE and HLA-C

通过 MHC-I 蛋白 HFE 和 HLA-C 的不同功能深入了解 PCSK9-LDLR 的调控和运输

Sepideh Mikaeeli, Ali Ben Djoudi Ouadda, Alexandra Evagelidis, Rachid Essalmani, Oscar Henrique Pereira Ramos, Carole Fruchart-Gaillard, Nabil G Seidah

Identification of PCPE-2 as the endogenous specific inhibitor of human BMP-1/tolloid-like proteinases

鉴定 PCPE-2 为人类 BMP-1/tolloid 样蛋白酶的内源性特异性抑制剂

Sandrine Vadon-Le Goff #, Agnès Tessier #, Manon Napoli #, Cindy Dieryckx, Julien Bauer, Mélissa Dussoyer, Priscillia Lagoutte, Célian Peyronnel, Lucie Essayan, Svenja Kleiser, Nicole Tueni, Emmanuel Bettler, Natacha Mariano, Elisabeth Errazuriz-Cerda, Carole Fruchart Gaillard, Florence Ruggiero, Ch

Molecular interactions of PCSK9 with an inhibitory nanobody, CAP1 and HLA-C: Functional regulation of LDLR levels.

PCSK9 与抑制性纳米抗体、CAP1 和 HLA-C 的分子相互作用:LDLR 水平的功能调节

Fruchart Gaillard Carole, Ouadda Ali Ben Djoudi, Ciccone Lidia, Girard Emmanuelle, Mikaeeli Sepideh, Evagelidis Alexandra, Le Dévéhat Maïlys, Susan-Resiga Delia, Lajeunesse Evelyne Cassar, Nozach Hervé, Ramos Oscar Henrique Pereira, Thureau Aurélien, Legrand Pierre, Prat Annik, Dive Vincent, Seidah Nabil G

New Hybrid Compounds Incorporating Natural Products as Multifunctional Agents against Alzheimer's Disease

含有天然产物的新型混合化合物可作为抗阿尔茨海默病的多功能药物

Lidia Ciccone, Caterina Camodeca, Nicolò Tonali, Lucia Barlettani, Armando Rossello, Carole Fruchart Gaillard, Julia Kaffy, Giovanni Petrarolo, Concettina La Motta, Susanna Nencetti, Elisabetta Orlandini

SKI-1/S1P Facilitates SARS-CoV-2 Spike Induced Cell-to-Cell Fusion via Activation of SREBP-2 and Metalloproteases, Whereas PCSK9 Enhances the Degradation of ACE2

SKI-1/S1P 通过激活 SREBP-2 和金属蛋白酶促进 SARS-CoV-2 刺突诱导的细胞间融合,而 PCSK9 则增强 ACE2 的降解

Rachid Essalmani, Ursula Andréo, Alexandra Evagelidis, Maïlys Le Dévéhat, Oscar Henrique Pereira Ramos, Carole Fruchart Gaillard, Delia Susan-Resiga, Éric A Cohen, Nabil G Seidah

Nature-Inspired O-Benzyl Oxime-Based Derivatives as New Dual-Acting Agents Targeting Aldose Reductase and Oxidative Stress

受自然启发的 O-苄基肟基衍生物作为针对醛糖还原酶和氧化应激的新型双作用药物

Lidia Ciccone, Giovanni Petrarolo, Francesca Barsuglia, Carole Fruchart-Gaillard, Evelyne Cassar Lajeunesse, Adeniyi T Adewumi, Mahmoud E S Soliman, Concettina La Motta, Elisabetta Orlandini, Susanna Nencetti

Copper mediated amyloid-β binding to Transthyretin

铜介导的β-淀粉样蛋白与转甲状腺素蛋白的结合

Ciccone, Lidia; Fruchart-Gaillard, Carole; Mourier, Gilles; Savko, Martin; Nencetti, Susanna; Orlandini, Elisabetta; Servent, Denis; Stura, Enrico A; Shepard, William

High throughput screening identifies disulfide isomerase DsbC as a very efficient partner for recombinant expression of small disulfide-rich proteins in E. coli

高通量筛选确定二硫键异构酶 DsbC 是大肠杆菌中重组表达富含二硫键的小蛋白质的非常有效的伙伴

Hervé Nozach, Carole Fruchart-Gaillard, François Fenaille, Fabrice Beau, Oscar Henrique Pereira Ramos, Badreddine Douzi, Natalie J Saez, Mireille Moutiez, Denis Servent, Muriel Gondry, Robert Thaï, Philippe Cuniasse, Renaud Vincentelli, Vincent Dive

Orthosteric binding of ρ-Da1a, a natural peptide of snake venom interacting selectively with the α1A-adrenoceptor

蛇毒天然肽 ρ-Da1a 的正构结合,与 α1A-肾上腺素能受体选择性相互作用

Arhamatoulaye Maïga, Jon Merlin, Elodie Marcon, Céline Rouget, Maud Larregola, Bernard Gilquin, Carole Fruchart-Gaillard, Evelyne Lajeunesse, Charles Marchetti, Alain Lorphelin, Laurent Bellanger, Roger J Summers, Dana S Hutchinson, Bronwyn A Evans, Denis Servent, Nicolas Gilles

Engineering of three-finger fold toxins creates ligands with original pharmacological profiles for muscarinic and adrenergic receptors

三指折叠毒素的工程设计产生了具有原始药理学特征的毒蕈碱和肾上腺素受体配体

Carole Fruchart-Gaillard, Gilles Mourier, Guillaume Blanchet, Laura Vera, Nicolas Gilles, Renée Ménez, Elodie Marcon, Enrico A Stura, Denis Servent