日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Quinazoline-Derivatives of Imino-1,2,3-Dithiazoles Promote Biofilm Dispersion of Pseudomonas aeruginosa

亚氨基-1,2,3-二噻唑的喹唑啉衍生物促进铜绿假单胞菌生物膜的分散

Gonzalez, Mathieu; Tareau, Anne-Sophie; de Crozals, Daphnée; Layec, Corentin; Broudic, Nathan; Barreau, Magalie; Forge, Adrien; Lesouhaitier, Olivier; Fruit, Corinne; Chevalier, Sylvie; Besson, Thierry; Tahrioui, Ali

Novel Thiazole-Fused [4,5-g] or [5,4-g]Quinazolin-8-ones and Their Quinazoline Analogues: Synthesis and Biological Evaluation.

新型噻唑稠合[4,5-g]或[5,4-g]喹唑啉-8-酮及其喹唑啉类似物:合成和生物学评价

Broudic Nathan, Pacheco-Benichou Alexandra, Corbière Cécile, Baratte Blandine, Robert Thomas, Bach Stéphane, Solhi Hélène, Le Guével Rémy, Fruit Corinne, Besson Thierry

Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts

利用二芳基碘鎓盐实现杂芳烃无过渡金属后期CH和NH芳基化反应的最新进展

Besson, Thierry; Fruit, Corinne

Development of Kinase Inhibitors via Metal-Catalyzed C⁻H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

通过片段增长研究设计的8-烷基噻唑并[5,4-f]喹唑啉-9-酮的金属催化C⁻H芳基化反应开发激酶抑制剂

Couly, Florence; Harari, Marine; Dubouilh-Benard, Carole; Bailly, Laetitia; Petit, Emilie; Diharce, Julien; Bonnet, Pascal; Meijer, Laurent; Fruit, Corinne; Besson, Thierry