日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Erratum for Dinh et al., "The structural and mechanistic bases for the viral resistance to allosteric HIV-1 integrase inhibitor pirmitegravir"

更正:Dinh 等人,“病毒对变构 HIV-1 整合酶抑制剂 pirmitegravir 产生耐药性的结构和机制基础”

Dinh, Tung; Tber, Zahira; Rey, Juan S; Mengshetti, Seema; Annamalai, Arun S; Haney, Reed; Briganti, Lorenzo; Amblard, Franck; Fuchs, James R; Cherepanov, Peter; Kim, Kyungjin; Schinazi, Raymond F; Perilla, Juan R; Kim, Baek; Kvaratskhelia, Mamuka

Delineating Structural Functionalities of Lenacapavir Amenable to Modifications for Targeting Emerging Drug-Resistant HIV‑1 Capsid Variants

阐明利那卡帕韦的结构功能,以便对其进行修饰,从而靶向新出现的耐药性 HIV-1 衣壳变体

Adu-Ampratwum, Daniel; Annamalai, Arun S; Dinh, Tung; Lockwood, Jeffrey R; Bockbrader, Ross H; Haney, Reed; Kvaratskhelia, Mamuka; Fuchs, James R

Additional Bioactive Silvestrol Analogs from the Roots of Aglaia perviridis Collected in Vietnam

从越南采集的绿叶阿格莱亚根中分离得到的其他生物活性西维斯醇类似物

Addo, Ermias Mekuria; Adu-Ampratwum, Daniel; Kaweesa, Elizabeth N; Agarwal, Garima; Uchenik, Dmitriy; Ninh, Tran N; Soejarto, Djaja D; Burdette, Joanna E; Fuchs, James R; Kinghorn, A Douglas; Rakotondraibe, Harinantenaina L

Antitumor and immunomodulatory activities of diphyllin and its derivatives

二氢槲皮素及其衍生物的抗肿瘤和免疫调节活性

Ren, Yulin; Gallucci, Judith C; Yu, Jianhua; Burdette, Joanna E; Fuchs, James R; Kinghorn, A Douglas

Verticillins: fungal epipolythiodioxopiperazine alkaloids with chemotherapeutic potential

维替西林:具有化学治疗潜力的真菌表多硫代二氧哌嗪生物碱

Pierre, Herma C; Amrine, Chiraz Soumia M; Doyle, Michael G; Salvi, Amrita; Raja, Huzefa A; Chekan, Jonathan R; Huntsman, Andrew C; Fuchs, James R; Liu, Kebin; Burdette, Joanna E; Pearce, Cedric J; Oberlies, Nicholas H

The structural and mechanistic bases for the viral resistance to allosteric HIV-1 integrase inhibitor pirmitegravir

病毒对变构HIV-1整合酶抑制剂吡米特格拉韦产生耐药性的结构和机制基础

Dinh, Tung; Tber, Zahira; Rey, Juan S; Mengshetti, Seema; Annamalai, Arun S; Haney, Reed; Briganti, Lorenzo; Amblard, Franck; Fuchs, James R; Cherepanov, Peter; Kim, Kyungjin; Schinazi, Raymond F; Perilla, Juan R; Kim, Baek; Kvaratskhelia, Mamuka

Semisynthetic derivatives of the fungal metabolite eupenifeldin via targeting the tropolone hydroxy groups

通过靶向托酚酮羟基合成真菌代谢物优培尼非林的半合成衍生物

Al Subeh, Zeinab Y; Pierre, Herma C; Bockbrader, Ross H; Tokarski, Robert J 2nd; Maldonado, Amanda C; Haughan, Monica A; Rangel-Grimaldo, Manuel E; Pearce, Cedric J; Burdette, Joanna E; Fuchs, James R; Oberlies, Nicholas H

Discovery and development of botanical natural products and their analogues as therapeutics for ovarian cancer

发现和开发植物天然产物及其类似物作为卵巢癌的治疗药物

Mize, Brittney K; Salvi, Amrita; Ren, Yulin; Burdette, Joanna E; Fuchs, James R

Efficacy of quorum sensing and growth inhibitors alone and in combination against avian pathogenic Escherichia coli infection in chickens

群体感应和生长抑制剂单独及联合应用对鸡禽致病性大肠杆菌感染的疗效

Helmy, Yosra A; Kathayat, Dipak; Closs, Gary Jr; Galgozy, Katie; Fuchs, James R; Rajashekara, Gireesh

Examination of the Impact of Triazole Position within Linkers on Solubility and Lipophilicity of a CDK9 Degrader Series

研究连接基团中三唑位置对 CDK9 降解剂系列溶解度和亲脂性的影响

Ayinde, Oluwatosin R; Sharpe, Chia; Stahl, Emily; Tokarski, Robert J 2nd; Lerma, James R; Muthusamy, Natarajan; Byrd, John C; Fuchs, James R