Discovery of a Potent and Selective ATAD2 Bromodomain Inhibitor with Antiproliferative Activity in Breast Cancer Models
发现一种在乳腺癌模型中具有抗增殖活性的强效选择性 ATAD2 溴结构域抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c01871
Jon J Winter-Holt, Catherine Bardelle, Elisabetta Chiarparin, Ian L Dale, Paul R J Davey, Nichola L Davies, Christopher Denz, Shaun M Fillery, Carine M Guérot, Fujin Han, Samantha J Hughes, Meghana Kulkarni, Zhaoqun Liu, Alexander Milbradt, Thomas A Moss, Huijun Niu, Joe Patel, Alfred A Rabow, Maria